Iferanserin

Name: Iferanserin
Brand: TargetMol
SKU: T15552
Rating: 4.5 (1 reviews)

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Catalog No. T15552Cas No. 58754-46-4

Alias S-MPEC

Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease.

Iferanserin

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Catalog No. T15552Alias S-MPECCas No. 58754-46-4

Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease.

Pack Size	Price	USA Warehouse	Global Warehouse
25 mg	$1,400	6-8 weeks	6-8 weeks
50 mg	$1,820	6-8 weeks	6-8 weeks
100 mg	$2,500	6-8 weeks	6-8 weeks

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Product Introduction

Bioactivity

Description	Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease.
In vitro	Iferanserin might modify the vascular effects occurring in hemorrhoid disease when it is used as an intra-anal ointment. Thereby decrease or eliminate the most frequently occurring symptoms of hemorrhoid disease[1].
Synonyms	S-MPEC

Chemical Properties

Molecular Weight	348.48
Formula	C₂₃H₂₈N₂O
Cas No.	58754-46-4
Relative Density.	1.096g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

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