Powder: -20°C for 3 years | In solvent: -80°C for 1 year
VER49009 (CCT0129397) is an effective HSP90 inhibitor(IC50 =25 nM, Kd=78 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 55.00 | |
2 mg | In stock | $ 77.00 | |
5 mg | In stock | $ 113.00 | |
10 mg | In stock | $ 176.00 | |
25 mg | In stock | $ 297.00 | |
50 mg | In stock | $ 497.00 | |
100 mg | In stock | $ 677.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 97.00 |
Description | VER49009 (CCT0129397) is an effective HSP90 inhibitor(IC50 =25 nM, Kd=78 nM). |
Targets&IC50 | HSP90:25 nM |
Kinase Assay | Fluorescence Polarization Assay: Binding of HSP90 inhibitors to human full-length recombinant HSP90β is determined by a competitive binding fluorescence polarization assay, using a fluorescent pyrazole resorcinol probe. |
Cell Research | Antiproliferative effects are measured using the sulforhodamine B assay. HUVEC sensitivity is determined by an alkaline phosphatase method. (Only for Reference) |
Synonyms | CCT0129397, VER 49009, VER-49009 |
Molecular Weight | 387.82 |
Formula | C19H18ClN3O4 |
CAS No. | 940289-57-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 71 mg/mL (183.1 mM)
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
VER49009 940289-57-6 Cytoskeletal Signaling Metabolism HSP CCT0129397 VER 49009 CCT 0129397 CCT-0129397 VER-49009 inhibitor inhibit