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Metabolism Phosphatase F1063-0967

F1063-0967

Catalog No. T4308   CAS 613225-56-2

F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11.62 μM.

F1063-0967, CAS 613225-56-2
Pack Size Availability Price/USD Quantity
1 mg In stock 27.00
2 mg In stock 36.00
5 mg In stock 54.00
10 mg In stock 86.00
50 mg In stock 230.00
100 mg In stock 320.00
1 mL * 10 mM (in DMSO) In stock 59.00
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Purity 99.15%
Biological Description
Chemical Properties
Storage & Solubility Information
Description F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11.62 μM.
Targets&IC50 DUSP26
Cell Research
The IMR-32 cells are plated in 96-well plates with 1×103 cells per well. After the cells are allowed to settle for 24 h, F1063-0967 (0, 10, 1, and 0.1 μM) is added. An MTTassay is performed. For cell lines HL7702 and SH-SY5Y, the cells are allowed to settle for 24 h, F1063-0967 (10 μM) is added, then MTT assays are carried out after 72 h.
Molecular Weight 484.59
Formula C24H24N2O5S2
CAS No. 613225-56-2

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

DMSO: 125 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Ren JX, et al. Identification of novel dual-specificity phosphatase 26 inhibitors by a hybrid virtual screening approach based on pharmacophore and molecular docking. Biomed Pharmacother. 2017 May;89:376-385.

Related compound libraries

This product is contained In the following compound libraries:
Bioactive Compound Library Inhibitor Library Anti-Metabolism Disease Compound Library Anti-cancer Metabolism Compound Library Phosphatase Inhibitor Library Covalent Inhibitor Library Lipid Metabolism Compound Library Glycometabolism Compound Library

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