Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).
Description | Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM). |
Targets&IC50 | D2 receptor:0.49 nM (ki), 5-HT1A receptor:2.6 nM (ki), D3 receptor:0.085 nM (ki) |
Molecular Weight | 413.38 |
Formula | C20H30Cl2N4O |
CAS No. | 839712-15-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Desmethyl cariprazine 839712-15-1 GPCR/G Protein Neuroscience Dopamine Receptor 5-HT Receptor inhibitor inhibit