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Cetilistat

Catalog No. T3283 CAS 282526-98-1

Synonyms: 新利司他, ATL-962

Cetilistat is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes.

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Cetilistat, CAS 282526-98-1

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Cetilistat is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes.
Targets&IC50	rat pancreatic lipase:54.8 nM, human pancreatic lipase:5.95 nM

Synonyms	新利司他, ATL-962
Molecular Weight	401.591
Formula	C25H39NO3
CAS No.	282526-98-1

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

H2O: Insoluble

DMSO: Insoluble

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Yamada Y et al. Hormone and Metabolic Research. 40 (8): 539–43.

Related Products

Related compounds with same targets

MAGL-IN-5 VK-28 Fatostatin PF 429242 Atractylodin Cetilistat Betulin Ethyl phenylglyoxylate

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Cetilistat 282526-98-1 代谢 Lipid ATL962 ATL-962 ATL 962 high-fat diet cholesterol Inhibitor anti-obesity pancreatic lipase inhibit inhibitor

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