keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Targefrin is a potent antagonist targeting EphA2, exhibiting a dissociation constant of 21 nM and an IC50 value of 10.8 nM for the EphA2-LBD. It promotes receptor internalization and degradation across multiple pancreatic cancer cell lines [1].
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Description | Targefrin is a potent antagonist targeting EphA2, exhibiting a dissociation constant of 21 nM and an IC50 value of 10.8 nM for the EphA2-LBD. It promotes receptor internalization and degradation across multiple pancreatic cancer cell lines [1]. |
Molecular Weight | 1700.94 |
Formula | C85H116F3N19O15 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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