Shopping Cart

Your shopping cart is currently empty

Lys-[Des-Arg9]Bradykinin,TFA

Name: Lys-[Des-Arg9]Bradykinin,TFA
Brand: TargetMol
SKU: TP1918L
Price: 47 USD
Availability: InStock
Rating: 5 (10 reviews)

Copy Product Info

🥰Excellent

Catalog No. TP1918L

Alias Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)

Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]-Bradykinin.

Lys-[Des-Arg9]Bradykinin,TFA

Copy Product Info

🥰Excellent

Purity: 97.35%

Catalog No. TP1918LAlias Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$47	In Stock	In Stock
5 mg	$107	In Stock	In Stock
10 mg	$161	In Stock	In Stock
25 mg	$289	In Stock	In Stock
50 mg	$413	In Stock	In Stock
100 mg	$589	In Stock	In Stock

Add to Cart

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:97.35%

Appearance:Solid

Color:White

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]-Bradykinin.
Synonyms	Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)

Chemical Properties

Molecular Weight	1260.24
Formula	C₅₄H₇₅F₆N₁₃O₁₅
Smiles	O=C(N1[C@H](C(NCC(N[C@@H](CC2=CC=CC=C2)C(N[C@H](C(N3[C@H](C(N[C@@H](CC4=CC=CC=C4)C(O)=O)=O)CCC3)=O)CO)=O)=O)=O)CCC1)[C@H]5N(C([C@@H](NC([C@H](CCCCN)N)=O)CCCNC(N)=N)=O)CCC5.OC(C(F)(F)F)=O.OC(C(F)(F)F)=O
Relative Density.	no data available
Sequence	H-Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-OH
Sequence Short	KRPPGFSPF

Storage & Solubility Information

Storage

keep away from moisture | Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 10 mM, Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	0.7935 mL	3.9675 mL	7.9350 mL	39.6750 mL
5 mM	0.1587 mL	0.7935 mL	1.5870 mL	7.9350 mL
10 mM	0.0793 mL	0.3967 mL	0.7935 mL	3.9675 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc