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d[Leu4,Lys8]-VP acetate

Catalog No. TP1927L1 CAS TP1927L1

Synonyms: d[Leu4,Lys8]-VP acetate(42061-33-6 free base)

d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4,Lys8]-VP acetate exhibits weak antidiuretic, vasopressor and oxytocic activiti

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d[Leu4,Lys8]-VP acetate, CAS TP1927L1

Pack Size	Availability	Price/USD
2 mg	In stock	$ 54.00
5 mg	In stock	$ 77.00
10 mg	In stock	$ 122.00
25 mg	In stock	$ 219.00
50 mg	In stock	$ 329.00
100 mg	In stock	$ 495.00
200 mg	In stock	$ 742.00
500 mg	In stock	$ 1,397.00

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Purity: 98.86%

Biological Description

Chemical Properties

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Description

Synonyms	d[Leu4,Lys8]-VP acetate(42061-33-6 free base)
Molecular Weight	1086.28
Formula	C49H71N11O13S2
CAS No.	TP1927L1

Storage

store at low temperture,keep away from moisture

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Ana P, et, al. Design and synthesis of the first selective agonists for the rat vasopressin V(1b) receptor: based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8. J Med Chem. 2007 Feb 22; 50(4): 835-47. 2. Ana P, et, al. Pharmacological and physiological characterization of d[Leu4, Lys8]vasopressin, the first V1b-selective agonist for rat vasopressin/oxytocin receptors. Endocrinology. 2007 Sep; 148(9): 4136-46.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Bioactive Compounds Library Max

Related Products

Related compounds with same targets

d[Leu4,Lys8]-VP acetate Argipressin LIXIVAPTAN Mozavaptan Desmopressin acetate (16679-58-6 free base) Desmopressin Atosiban Fuscoside

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

d[Leu4,Lys8]-VP acetate TP1927L1 GPCR/G Protein Vasopressin Receptor d[Leu4,Lys8]VP acetate d[Leu4,Lys8]-VP acetate(42061-33-6 free base) d[Leu4,Lys8] VP acetate Inhibitor inhibitor inhibit

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