Powder: -20°C for 3 years | In solvent: -80°C for 1 year
NTRC-824 is <150-fold selectivity for NTS2 over NTS1 (Ki <30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
50 mg | 35 days | $ 3,510.00 |
Description | NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM). |
Targets&IC50 | NTS2:(ki)202 nM, NTS2:38 nM |
In vitro | NTRC-824 is the first nonpeptide compound that behaves like and is more active than, the endogenous ligand. In the NTS1 assay up to 30 μM, Testing of NTRC-824 at the NTS1 receptor displays no binding activity, making NTRC-824 selective for NTS2 in both the binding and functional assays . |
Molecular Weight | 553.55 |
Formula | C25H26F3N3O6S |
CAS No. | 1623002-61-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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NTRC-824 1623002-61-8 Others NTRC824 NTRC 824 inhibitor inhibit