store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits the growth of cancer cells.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 854.00 | |
50 mg | 8-10 weeks | $ 1,110.00 | |
100 mg | 8-10 weeks | $ 1,680.00 |
Description | KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits the growth of cancer cells. |
Targets&IC50 | c-Src:86 nM (Kd), c-Src:44 nM (Ki) |
In vitro | KB SRC 4 is a highly selective c-Src inhibitor. The Kd for c-Src (86 nM) is consistent with the Ki obtained in our biochemical activity assay. Compound 4(KB SRC 4) exhibits selectivity among Src family members, with >2-fold selectivity over both Lck and Fgr, 8-fold selectivity over c-Yes, and >40-fold selectivity over Lyn, Hck, and Fyn.[1]. |
Molecular Weight | 555.03 |
Formula | C32H23ClN8 |
CAS No. | 1380088-03-8 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 80 mg/mL (144.14 mM), sonification is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
KB SRC 4 1380088-03-8 Angiogenesis Tyrosine Kinase/Adaptors Src inhibitor inhibit