Powder: -20°C for 3 years | In solvent: -80°C for 1 year
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors. |
In vitro | (E)-GABAB receptor antagonist 1 ?decreases agonist GABA-induced maximal effect of IP3 production in HEK293 cells overexpressing GABAB receptors and Gqi9 proteins without changing the EC50. |
Molecular Weight | 304.38 |
Formula | C18H24O4 |
CAS No. | 797-17-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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GABAB receptor antagonist 1 797-17-1 Membrane transporter/Ion channel Neuroscience GABA Receptor inhibitor inhibit