Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 213.00 | |
5 mg | In stock | $ 537.00 | |
10 mg | In stock | $ 775.00 | |
25 mg | In stock | $ 1,190.00 | |
50 mg | In stock | $ 1,590.00 | |
100 mg | In stock | $ 2,170.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 593.00 |
Description | ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively. |
Targets&IC50 | ERK2:3.0 nM, ERK1: |
In vitro | ERK1/2 inhibitor 1 ?shows excellent antiproliferative potency with IC50s of 7.5 and 4.9 nM in ?Colo205 cells and A375, respectively. |
Molecular Weight | 550.05 |
Formula | C29H32ClN5O4 |
CAS No. | 2095719-90-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.5 mg/mL (10 mM), Sonification is recommended
You can also refer to dose conversion for different animals. More
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ERK1/2 inhibitor 1 2095719-90-5 MAPK ERK ERK-1/2 inhibitor 1 inhibitor inhibit