Shopping Cart
- Remove All
![TargetMol](https://www.targetmol.com/storage/error/oops.webp)
Your shopping cart is currently empty
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,820 | 8-10 weeks | |
50 mg | $2,380 | 8-10 weeks | |
100 mg | $3,100 | 8-10 weeks |
Description | CCT251455 is an inhibitor of mitotic kinase monopolar spindle 1 (MPS1; IC50: 3 nM). |
In vitro | CCT251455 is a highly potent inhibitor of MPS1 that demonstrates high selectivity versus kinases tested in a broad kinome profiling panel. CCT251455 inhibits P-MPS1 (IC50: 0.04 μM in the cell-based assay; GI50: 0.16 μM). |
In vivo | CCT251455 demonstrates a good oral pharmacokinetic profile in mice and rats as well as inhibition of MPS1 activity in vivo following oral administration. |
Molecular Weight | 503.98 |
Formula | C26H26ClN7O2 |
Cas No. | 1400284-80-1 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.