Shopping Cart
- Remove All
Your shopping cart is currently empty
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
🥰Excellent
Catalog No. TP1893L1
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively) and displays anti-inflammatory efficacy.
![[D-Trp8]-γ-MSH acetate(321351-81-9 free base)](/group3/M00/12/DA/CgoaEGZGsH2Eawr8AAAAAM5W_vs327.png)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
🥰Excellent
Purity: 100%
Catalog No. TP1893L1
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively) and displays anti-inflammatory efficacy.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 135 € | In Stock | |
| 5 mg | 306 € | In Stock | |
| 10 mg | 443 € | In Stock | |
| 25 mg | 672 € | In Stock | |
| 50 mg | 905 € | In Stock | |
| 100 mg | 1.235 € | In Stock | |
| 200 mg | 1.672 € | In Stock |
Bulk & Custom
Add to Cart
Questions
View MoreInhibitors Related to "[D-Trp8]-γ-MSH acetate(321351-81-9 free base)"
Bremelanotide Acetate
PT-141 Acetate
T76081607799-13-2
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
- 43 €
Size
QTY
Fenoprofen
Nalgesic, Nalfon
T0184L29679-58-1
Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, which increases ERK1/2 activation, inhibits biofilm formation, and alters biofilm structure, and is used in the treatment of acute pain and chronic arthritis.
- 28 €
Size
QTY
HS024
HS 024
TP1898212370-59-7
HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.
- 328 €
Size
QTY
ACTH 11-24 acetate(4237-93-8 free base)
Adrenocorticotropic Hormone (11-24) acetate
TP1248L79190-56-0
ACTH 11-24 acetate(4237-93-8 free base) (Adrenocorticotropic Hormone (11-24) acetate) is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39) and ACTH (1-10) in isolated adrenal cells.
- 41 €
Size
QTY
Undecylenoyl phenylalanine
Undecylenoylphenylalanine, Sepiwhite msh QD
T20501175357-18-3
Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an alpha-melanocyte-stimulating hormone antagonist, thus inhibiting melaninogenesis.
- 27 €
Size
QTY
Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt, Melanostatine-5 acetate salt
TP1101
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt (158563-45-2 free base) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM.
- 59 €
Size
QTY
Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate(125934-45-4 free base)
TP1578L
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
- 61 €
Size
QTY
BMS-470539 dihydrochloride
BMS470539 dihydrochloride, BMS 470539 dihydrochloride
T105682341796-82-3
BMS-470539 dihydrochloride is a selective and highly potent melanocortin 1 receptor (MC-1 R) agonist with anti-inflammatory activity. BMS-470539 attenuates oxidative stress and neuronal apoptosis via the MC1R/cAMP/PKA/Nurr1 signaling pathway in a neonatal hypoxia-ischemia rat model.
- 49 €
Size
QTY
ACTH (1-17) acetate
TP1011L
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
- 115 €
Size
QTY
Beta-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)
TP1004L
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.
- 158 €
Size
QTY
MCL0020
MCL 0020
TP1889475498-26-1
MCL0020 is a potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115, and >10,000 nM at MC4, MC3, and MC1 receptors, respectively). It significantly reverses stress-induced anorexia without affecting food intake in free-feeding rats and exhibits anxiolytic-like activity in vivo.
- 112 €
Size
QTY
HS 014 acetate(207678-81-7 free base)
TP2015L
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake in rats and nociception in mice following central
- 175 €
Size
QTY
Select Batch
Purity:100%
Contact us for more batch information
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | [D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively) and displays anti-inflammatory efficacy. |
| Targets&IC50 | MC3:6.7 Nm, MC5R:340 Nm, MC4R:600 nM |
| Molecular Weight | 1630.82 |
| Formula | C76H103N21O18S |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | H2O: Insoluble DMSO: Insoluble |
Sci Citations
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
Keywords
MelanocortinReceptormelanocortin-5 receptor (MC5R)melanocortin-4 receptor (MC4R)Melanocortin Receptormelanocortin 3 (MC3)[D-Trp8]-γ-MSH acetate(321351-81-9 free base)[D-Trp-8]-γ-MSH acetate(321351-81-9 free base)[DTrp8]γMSH acetate(321351819 free base)[D-Trp8]-r-MSH acetate(321351-81-9 free base)[D-Trp8]-gamma-MSH acetate(321351-81-9 free base)[D Trp8] γ MSH acetate(321351 81 9 free base)
Preview
Related Tags: buy [D-Trp8]-γ-MSH acetate(321351-81-9 free base) | purchase [D-Trp8]-γ-MSH acetate(321351-81-9 free base) | [D-Trp8]-γ-MSH acetate(321351-81-9 free base) cost | order [D-Trp8]-γ-MSH acetate(321351-81-9 free base) | [D-Trp8]-γ-MSH acetate(321351-81-9 free base) chemical structure | [D-Trp8]-γ-MSH acetate(321351-81-9 free base) formula | [D-Trp8]-γ-MSH acetate(321351-81-9 free base) molecular weight
- TOP
Feedback
Hello! How can I help you today? 
Copyright © 2015-2025 TargetMol Chemicals Inc. All Rights Reserved.