keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat brain in vitro (IC50 = 3 - 15 nM). Attenuates the antidepressant effects of fluoxetine and blocks galanin-induced food intake in vivo. Also exhibits weak partial agonist activity at peripheral GAL2 receptors at doses < 100 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 196.00 | |
5 mg | In stock | $ 487.00 | |
10 mg | In stock | $ 696.00 | |
25 mg | In stock | $ 1,090.00 | |
50 mg | In stock | $ 1,490.00 | |
100 mg | In stock | $ 1,980.00 |
Description | M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat brain in vitro (IC50 = 3 - 15 nM). Attenuates the antidepressant effects of fluoxetine and blocks galanin-induced food intake in vivo. Also exhibits weak partial agonist activity at peripheral GAL2 receptors at doses > 100 nM. |
Molecular Weight | 2041.38 |
Formula | C96H149N23O26 |
CAS No. | TP1992L |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10 mM
You can also refer to dose conversion for different animals. More
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M40 acetate(143896-17-7 free base) TP1992L GPCR/G Protein Neuroscience Neuropeptide Y Receptor M-40 acetate(143896-17-7 free base) M40 acetate(143896 17 7 free base) M40 acetate(143896177 free base) inhibitor inhibit