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L 365209

Catalog No. T24288 CAS 122211-30-7

Synonyms: L365,209, L365209, L 365,209, L-365,209, L-365209

L 365209 is an oxytocin antagonist.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

L 365209, CAS 122211-30-7

Pack Size	Availability	Price/USD
25 mg	10-14 weeks	$ 3,620.00
50 mg	10-14 weeks	$ 4,780.00
100 mg	10-14 weeks	$ 6,700.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description

L 365209 is an oxytocin antagonist.

Synonyms	L365,209, L365209, L 365,209, L-365,209, L-365209
Molecular Weight	738.88
Formula	C40H50N8O6
CAS No.	122211-30-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Geenen V, Martens H, Robert F, Vrindts-Gevaert Y, De Groote D, Franchimont P. Immunomodulatory properties of cyclic hexapeptide oxytocin antagonists. Thymus. 1992 Dec;20(4):217-26. PubMed PMID: 1492361. 2. Williams PD, Bock MG, Tung RD, Garsky VM, Perlow DS, Erb JM, Lundell GF, Gould NP, Whitter WL, Hoffman JB, et al. Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product. J Med Chem. 1992 Oct 16;35(21):3905-18. PubMed PMID: 1331448. 3. Pettibone DJ, Clineschmidt BV, Lis EV, Reiss DR, Totaro JA, Woyden CJ, Bock MG, Freidinger RM, Tung RD, Veber DF, et al. In vitro pharmacological profile of a novel structural class of oxytocin antagonists. J Pharmacol Exp Ther. 1991 Jan;256(1):304-8. PubMed PMID: 1988661. 4. Grider JR, Makhlouf GM. Distinct receptors for cholecystokinin and gastrin on muscle cells of stomach and gallbladder. Am J Physiol. 1990 Aug;259(2 Pt 1):G184-90. PubMed PMID: 2382717.

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

L 365209 122211-30-7 L365,209 L365209 L 365,209 L-365,209 L-365209 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.