Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
Description | GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions. |
Targets&IC50 | A1 receptor:3.1 nM (cell free) |
In vivo | GR79236 has been shown to have antinociceptive and anti-inflammatory properties in animal models. GR79236 inhibits the release of CGRP evoked by superior sagittal sinus (SSS) stimulation in the cat and inhibits trigeminal nucleus firing in the cat and rat. GR79236X has acute, short-term analgesic efficacy. |
Synonyms | GR 79236 |
Molecular Weight | 351.36 |
Formula | C15H21N5O5 |
CAS No. | 124555-18-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 98 mg/mL (278.92 mM)
You can also refer to dose conversion for different animals. More
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GR79236 124555-18-6 GPCR/G Protein Neuroscience Adenosine Receptor GR-79236 GR 79236 inhibitor inhibit