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AC 187 Acetate

Catalog No. T21581L CAS T21581L

Synonyms: AC 187 Acetate (151804-77-2 Free base)

AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.

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AC 187 Acetate, CAS T21581L

Pack Size	Availability	Price/USD
1 mg	In stock	$ 917.00
5 mg	In stock	$ 1,860.00
10 mg	In stock	$ 2,480.00
25 mg	In stock	$ 3,720.00
50 mg	In stock	$ 4,920.00
100 mg	In stock	$ 6,770.00

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Purity: 99.71%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.
Targets&IC50	Amylin receptor:0.48 nM
In vitro	AC187 attenuates the activation of initiator and effector caspases that mediate Aβ-induced apoptotic cell death.

Synonyms	AC 187 Acetate (151804-77-2 Free base)
Molecular Weight	2950.26
Formula	C129H209N37O42
CAS No.	T21581L

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 90 mg/mL (29.96 mM), Sonication is recommended.

References and Literature

1. Jack H Jhamandas, et al. Antagonist of the amylin receptor blocks beta-amyloid toxicity in rat cholinergic basal forebrain neurons. J Neurosci. 2004 Jun 16;24(24):5579-84.

Related compound libraries

This product is contained In the following compound libraries：

NO PAINS Compound Library Natural Product Library for HTS Natural Product Library

Related Products

Related compounds with same targets

Amylin, amide, rat acetate(124447-81-0,free base) cAC 253 acetate

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Keywords

AC 187 Acetate T21581L GPCR/G Protein Amylin Receptor AC-187 Acetate 151804-77-2 AC187 Acetate 151804-77-2 Free base AC 187 Acetate (151804-77-2 Free base) inhibitor inhibit

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