Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ITI-214 free base is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
50 mg | 8-10 weeks | $ 789.00 | |
100 mg | 8-10 weeks | $ 1,180.00 |
Description | ITI-214 free base is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). |
Targets&IC50 | PDE1C:35 pM (Ki), PDE1A:33 pM (Ki), PDE1B:380 pM (Ki), PDE1:58 pM (Ki) |
Synonyms | ITI214 free base |
Molecular Weight | 507.56 |
Formula | C29H26FN7O |
CAS No. | 1160521-50-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
ITI-214 free base 1160521-50-5 Others ITI214 ITI214 free base ITI-214 ITI 214 ITI 214 free base inhibitor inhibit