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Clobenpropit 2HBr

Catalog No. T19762 CAS 145231-45-4

Synonyms: VUF-9153, VUF 9153, Clobenpropit Dihydrobromide, VUF9153

Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.

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Clobenpropit 2HBr, CAS 145231-45-4

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.

Synonyms	VUF-9153, VUF 9153, Clobenpropit Dihydrobromide, VUF9153
Molecular Weight	308.83
Formula	C14H17ClN4S
CAS No.	145231-45-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: Soluble

References and Literature

1. Schneider E, Bertron AF, Dy M. Modulation of hematopoiesis through histamine receptor signaling. Front Biosci (Schol Ed). 2011 Jan 1;3:467-73. Review. PubMed PMID: 21196390. 2. Bleicher KH, Green LG, Martin RE, Rogers-Evans M. Ligand identification for G-protein-coupled receptors: a lead generation perspective. Curr Opin Chem Biol. 2004 Jun;8(3):287-96. Review. PubMed PMID: 15183327. 3. Oda T, Matsumoto S. [Identification and characterization of histamine H4 receptor]. Nihon Yakurigaku Zasshi. 2001 Jul;118(1):36-42. Review. Japanese. PubMed PMID: 11496825. 4. Kamei C, Okuma C. [Role of central histamine in amygdaloid kindled seizures]. Nihon Yakurigaku Zasshi. 2001 May;117(5):329-34. Review. Japanese. PubMed PMID: 11411342.

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Clobenpropit 2HBr 145231-45-4 Clobenpropit VUF-9153 VUF 9153 Clobenpropit Dihydrobromide VUF9153 inhibitor inhibit

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