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BMY-25271

Catalog No. T10575 CAS 78441-82-4

BMY-25271 is an antagonist of histamine H2 receptor.

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BMY-25271, CAS 78441-82-4

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description	BMY-25271 is an antagonist of histamine H2 receptor.
In vivo	The dose-response curves are parallel and oral ED50 values derived from probit analysis are 0.093, 0.97, and 6.9 mg/kg for BMY-25271, ranitidine, and cimetidine, respectively. BMY-25271 is about 10 and 74 times more potent than ranitidine and cimetidine, respectively.

Molecular Weight	329.44
Formula	C12H19N5O2S2
CAS No.	78441-82-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Cavanagh RL, et al. Prevention of aspirin-induced gastric mucosal injury by histamine H2 receptor antagonists: a crossover endoscopic and intragastric pH study in the dog. J Pharmacol Exp Ther. 1987 Dec;243(3):1179-84.

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Mequitazine Lodoxamide tromethamine JNJ-7777120 Bavisant Imetit dihydrobromide LY-2624803 Cimetidine Samelisant

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

BMY-25271 78441-82-4 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor BMY 25271 BMY25271 inhibitor inhibit

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