keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
JKC363 TFA is a selective melanocortin MC4 receptor antagonist that exhibits a 90-fold higher affinity for the MC4 receptor (IC50=0.5 nM) compared to the MC3 receptor (44.9 nM). This compound effectively inhibits the α-MSH-induced stimulation of TRH release. It also demonstrates an anti-hyperalgesic effect [1] [2].
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Description | JKC363 TFA is a selective melanocortin MC4 receptor antagonist that exhibits a 90-fold higher affinity for the MC4 receptor (IC50=0.5 nM) compared to the MC3 receptor (44.9 nM). This compound effectively inhibits the α-MSH-induced stimulation of TRH release. It also demonstrates an anti-hyperalgesic effect [1] [2]. |
Molecular Weight | 1620.73 |
Formula | C71H93F3N19O18S2 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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