[D-Trp2,7,9] Substance P

Name: [D-Trp2,7,9] Substance P
Brand: TargetMol
SKU: T76405
Rating: 4.5 (1 reviews)

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Catalog No. T76405Cas No. 100930-11-8

[D-Trp2,7,9] Substance P is a tachykinin (Neurokinin Receptor) antagonist with inhibitory affinities (K_i values) of 1 μM for NK-1, 1.3 μM for NK-2, and approximately 9 μM for NK-3 receptors [1].

[D-Trp2,7,9] Substance P

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Catalog No. T76405Cas No. 100930-11-8

[D-Trp2,7,9] Substance P is a tachykinin (Neurokinin Receptor) antagonist with inhibitory affinities (K_i values) of 1 μM for NK-1, 1.3 μM for NK-2, and approximately 9 μM for NK-3 receptors [1].

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Product Introduction

Bioactivity

Description	[D-Trp2,7,9] Substance P is a tachykinin (Neurokinin Receptor) antagonist with inhibitory affinities (K_i values) of 1 μM for NK-1, 1.3 μM for NK-2, and approximately 9 μM for NK-3 receptors [1].
Targets&IC50	NK2:1.3 μM (Ki), NK3:~9 μM (Ki), NK1:1 μM (Ki)

Chemical Properties

Molecular Weight	1604.92
Formula	C₈₀H₁₀₉N₂₁O₁₃S
Cas No.	100930-11-8
Sequence Short	RWKPQQWFWLM-NH2

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

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