Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2 nM and induces vasoconstriction in rabbit pulmonary arteries. Additionally, it promotes relaxation of the pig urinary bladder neck, rendering it useful for research into cardiovascular diseases [1] [2].
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Description | BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2 nM and induces vasoconstriction in rabbit pulmonary arteries. Additionally, it promotes relaxation of the pig urinary bladder neck, rendering it useful for research into cardiovascular diseases [1] [2]. |
Molecular Weight | 2006.32 (free base) |
Formula | C96H140N20O25S.xNH3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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BQ-3020 ammonium GPCR/G Protein Endothelin Receptor inhibitor inhibit