Powder: -20°C for 3 years | In solvent: -80°C for 1 year
TAK1/MAP4K2 inhibitor 1 is a potent dual inhibitor of TGFβ-activated kinase 1 (TAK1) and MAP4K2 (IC50s: 41.1 nM and 18.2 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | 5 days | $ 177.00 | |
5 mg | 5 days | $ 297.00 | |
25 mg | 6-8 weeks | $ 766.00 | |
50 mg | 6-8 weeks | $ 996.00 | |
100 mg | 6-8 weeks | $ 1,590.00 | |
1 mL * 10 mM (in DMSO) | 5 days | $ 372.00 |
Description | TAK1/MAP4K2 inhibitor 1 is a potent dual inhibitor of TGFβ-activated kinase 1 (TAK1) and MAP4K2 (IC50s: 41.1 nM and 18.2 nM). |
Targets&IC50 | MAP4K2:18.2 nM, TAK1:41.1 nM |
In vivo | TAK1/MAP4K2 inhibitor 1 (1 mg/kg, iv) has moderate terminal elimination half-life (t1/2=2.94 h) in mice. |
Molecular Weight | 552.59 |
Formula | C29H31F3N6O2 |
CAS No. | 1315330-11-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (90.48 mM), sonification is recommended.
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
TAK1/MAP4K2 inhibitor 1 1315330-11-0 Others TAK-1/MAP4K2 inhibitor 1 inhibitor inhibit