Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM, exhibits < 200-fold selectivity over other HDAC.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 57.00 | |
10 mg | In stock | $ 82.00 | |
25 mg | In stock | $ 136.00 | |
50 mg | In stock | $ 202.00 | |
100 mg | In stock | $ 303.00 |
Description | RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM, exhibits > 200-fold selectivity over other HDAC. |
Targets&IC50 | HDAC3:0.08 μM |
In vitro | In mammals, halofuginone at 10 ng/ml down-regulates Smad3, blocking TGF-β signaling and preventing both the differentiation of fibroblasts to myofibroblasts and the transitioning of epithelial cells to mesenchymal cells[2]. |
Molecular Weight | 362.4 |
Formula | C21H19FN4O |
CAS No. | 1396841-57-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
H2O: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 67 mg/mL (184.9 mM)
You can also refer to dose conversion for different animals. More
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RGFP966 (E-isomer) 1396841-57-8 Chromatin/Epigenetic DNA Damage/DNA Repair HDAC E-isomer RGFP-966 RGFP 966 RGFP966 inhibitor inhibit