Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin-converting enzyme (ACE) inhibitor (IC50: 2.6 nM). It is used in the research of the hypertensive disease.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
500 μg | 35 days | $ 398.00 | |
1 mg | 35 days | $ 715.00 |
Description | Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin-converting enzyme (ACE) inhibitor (IC50: 2.6 nM). It is used in the research of the hypertensive disease. |
Targets&IC50 | ACE:2.6 nM |
In vitro | Imidaprilate augments the bradykinin-induced contraction of guinea pig ileum, with AC50 of 1.7 nM.Imidaprilate ?is an active metabolite of 6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM. |
In vivo | Imidaprilate (≥0.2 mg/kg) inhibits angiotensin I (AT-I)-induced pressor response. |
Synonyms | Imidaprilat, 6366A |
Molecular Weight | 377.39 |
Formula | C18H23N3O6 |
CAS No. | 89371-44-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Imidaprilate 89371-44-8 Endocrinology/Hormones RAAS Imidaprilat 6366A inhibitor inhibit