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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
NF-κB
CDK
Dopamine Receptor
COX
PI3K
Antibacterial
Adrenergic Receptor
AChR
EGFR
HIV Protease
Potassium Channel
VEGFR
DNA/RNA Synthesis
Cytochromes P450
Calcium Channel
Antibiotic
Histamine Receptor
Reactive Oxygen Species
TNF
Akt
Epigenetic Reader Domain
ERK
Sodium Channel
JAK
mTOR
Estrogen/progestogen Receptor
FLT
PDGFR
Src
PDE
PPAR
Dehydrogenase
Ferroptosis
HDAC
IL Receptor
p38 MAPK
Parasite
FGFR
Histone Methyltransferase
iGluR
PKC
c-Kit
Influenza Virus
STAT
Wnt/beta-catenin
TRP/TRPV Channel
Caspase
Estrogen Receptor/ERR
SARS-CoV
GABA Receptor
PARP
AMPK
Bcl-2 Family
NO Synthase
GSK-3
Microtubule Associated
NMDAR
ALK
MMP
GluR
c-Met/HGFR
ROS
Bcr-Abl
MAO
Cholinesterase (ChE)
Raf
Antifungal
MAPK
Prostaglandin Receptor
Virus Protease
Aurora Kinase
Mitophagy
Topoisomerase
Tyrosine Kinases
TLR
HSV
Phosphatase
JNK
Ras
Beta Amyloid
Proteasome
HCV Protease
HIF/HIF Prolyl-Hydroxylase
HSP
Lipoxygenase
TGF-beta/Smad
ATPase
MEK
Cannabinoid Receptor
Casein Kinase
GPCR
Norepinephrine
p53
Interleukin
PKA
Adenosine Receptor
Mitochondrial Metabolism
Sirtuin
Monoamine Oxidase
Reverse Transcriptase
ROCK
Antiviral
E1/E2/E3 Enzyme
Nrf2
P-gp
IκB/IKK
NOS
RAAS
TAM Receptor
Drug Metabolite
LPL Receptor
Phospholipase
S6 Kinase
Serotonin Transporter
Glucocorticoid Receptor
IGF-1R
DNA-PK
HIF
Retinoid Receptor
S1P Receptor
Serine/threonin kinase
HER
Antioxidant
c-RET
Gamma-secretase
Carbonic Anhydrase
DUB
Trk receptor
Androgen Receptor
HBV
Opioid Receptor
Integrin
Nucleoside Antimetabolite/Analog
Serine Protease
Cysteine Protease
Progesterone Receptor
Histone Demethylase
Mdm2
Tyrosinase
c-Fms
Histone Acetyltransferase
NOD
Pim
Rho
CaMK
CCR
FAK
HMG-CoA Reductase
PERK
ATM/ATR
BACE
CXCR
DNA Alkylator/Crosslinker
DYRK
Hedgehog/Smoothened
Syk
Transferase
DNA Methyltransferase
MRP
PLK
PROTACs
Chk
DPP-4
Sigma receptor
transporter
Aryl Hydrocarbon Receptor
NADPH
NOD-like Receptor (NLR)
P2X Receptor
RIP kinase
Smo
Acyltransferase
AhR
Chloride channel
Fatty Acid Synthase
Glucosidase
Glutathione Peroxidase
Proton pump
Beta-Secretase
DNA
DNA Alkylation
FAAH
Indoleamine 2,3-Dioxygenase (IDO)
CSF-1R
Immunology/Inflammation related
PAK
PDK
ROS Kinase
ABC Transporter
Antifection
cAMP
IAP
Kinesin
LDL
LTR
Reductase
Stearoyl-CoA Desaturase (SCD)
Thrombin
GPCR19
IRAK
P2Y Receptor
SGLT
ADC Cytotoxin
c-Myc
Isocitrate Dehydrogenase (IDH)
Liver X Receptor
LPA Receptor
MNK
PGE Synthase
YAP
DHFR
Endothelin Receptor
FXR
IDO
Leukotriene Receptor
LRRK2
MT Receptor
UGT
Antifolate
Aromatase
BTK
CFTR
Discoidin Domain Receptor (DDR)
DNA gyrase
Epoxide Hydrolase
GTPase
IFNAR
Lipid
Melatonin Receptor
Myosin
OX Receptor
PI4K
ribosome
Xanthine Oxidase
Amino Acids and Derivatives
Anti-infection
BCRP
Ephrin Receptor
Free radical scavengers
GST
Ligands for Target Protein for PROTAC
LIM Kinase
MLK
Monoamine Transporter
NADPH-oxidase
PD-1/PD-L1
PYK2
ROR
SGK
STING
Telomerase
Thyroid hormone receptor(THR)
Vasopressin Receptor
Aminopeptidase
Arginase
CRISPR/Cas9
Guanylate cyclase
Lipase
MicroRNA
PAFR
Platelet aggregation
SIK
Tie-2
Annexin A
ASK
Complement System
Factor Xa
Glucagon Receptor
Glucokinase
GPX
Imidazoline Receptor
NAMPT
Neurokinin receptor
Phosphorylase
Protease-activated Receptor
PTEN
RSV
AAK1
ACK1
Arrestin
ATP Citrate Lyase
Carboxypeptidase
Decarboxylase
Dynamin
GRK
Hydroxylase
IRE1
MTH1
MyD88
Na+/Ca2+ Exchanger
NPC1L1
OAT
PAI-1
Porcupine
Pyroptosis
RAR/RXR
Kras
Adenosine Deaminase
Adenylyl Cyclase
AIM2
Amylase
cGAS
Cholecystokinin Receptor
Gap Junction Protein
GHSR
GluCls
Glutaminase
GlyT
Hck
Hexokinase
Ligand for E3 Ligase
MAGL
Melanin-concentrating Hormone Receptor (MCHR)
Melanocortin Receptor
Molecular Glues
NEDD8
Neuropeptide Y Receptor
PAD
Thrombopoietin Receptor
TOPK
Transaminase
FOXO3
Adiponectin Receptor
Advanced Glycation End Products
BMI-1
Bombesin Receptor
Cell Cycle Arrest
CGRP Receptor
CPT
CRFR
CRM1
DAPK
FLAP
Glutathione reductase
GNRH Receptor
gp120/CD4
Haspin Kinase
Hippo pathway
Huntingtin
KLF
KSP
Lysosomal Autophagy
MELK
Monocarboxylate transporter
Neprilysin
OCT
OXPHOS
Oxytocin Receptor
PKM
Protease
VDA
Wee1
IKZF
Acetyl-CoA Carboxylase
Aconitase
Angiotensin-converting Enzyme (ACE)
Anion Exchanger
APC/C
Aquaporin
ATTECs
CaSR
Cell wall
CETP
EBI2/GPR183
FABP
Fas/FasL
GSNOR
hCE
HCN Channel
Integrase
Methionine Adenosyltransferase (MAT)
N-Acetylglucosaminyltransferase
Na-K-Cl cotransporter
Necroptosis
p97
PROTAC Linker
RANKL/RANK
RXFP receptor
Somatostatin
Survivin
Taste receptor

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