keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
TAK-448 acetate (MVT-602 acetate) is a small molecule KISS1R agonist, a synthetic peptide similar to kisspeptin.TAK-448 acetate has antitumor activity, inhibits the proliferation of VCaP cells, and can be used in prostate cancer research.TAK-448 acetate is a small molecule KISS1R agonist.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 121.00 | |
5 mg | In stock | $ 247.00 | |
10 mg | In stock | $ 396.00 | |
25 mg | In stock | $ 648.00 | |
50 mg | In stock | $ 929.00 |
Description | TAK-448 acetate (MVT-602 acetate) is a small molecule KISS1R agonist, a synthetic peptide similar to kisspeptin.TAK-448 acetate has antitumor activity, inhibits the proliferation of VCaP cells, and can be used in prostate cancer research.TAK-448 acetate is a small molecule KISS1R agonist. |
Targets&IC50 | KISS1R:632 pM, KISS1R:460 pM |
In vivo | A single injection of TAK-448 significantly increases plasma levels of follicle-stimulating hormone and testosterone (T) in male rats. In the androgen-sensitive prostate cancer model of male rats with VCaP xenografts, TAK-448 (0.01, 0.03, 0.3, 3 mg/kg; i.h.; 0,28 days) exhibits greater anti-tumor effects[1]. |
Synonyms | TAK-448 acetate (1234319-68-6 Free base), MVT-602 acetate |
Molecular Weight | 1285.41 |
Formula | C60H84N16O16 |
CAS No. | 1470374-22-1 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 80 mg/mL (62.24 mM), Sonication is recommended.
H2O: 30 mg/mL (23.34 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
TAK-448 acetate 1470374-22-1 GPCR/G Protein Kisspeptin TAK-448 acetate (1234319-68-6 Free base) TAK-448 Acetate MVT 602 Acetate MVT-602 acetate MVT602 Acetate inhibitor inhibit