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TOPRelated productsBioactivityChemical infoStorage&SolubilityCalculator

PKI (5-24) Acetate(99534-03-9 free base)

🥰Excellent
Catalog No. TP1957L

PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM).

PKI (5-24) Acetate(99534-03-9 free base)
Other Forms of PKI (5-24) Acetate(99534-03-9 free base):
PKI(5-24)TP195799534-03-9
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PKI (5-24) Acetate(99534-03-9 free base)

🥰Excellent
Purity: 99.47%
Catalog No. TP1957L
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM).
Pack SizePriceAvailabilityQuantity
1 mg$79In Stock
5 mg$162In Stock
10 mg$273In Stock
25 mg$452In Stock
50 mg$636In Stock
100 mg$858In Stock
200 mg$1,150In Stock
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Purity:99.47%
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COA MS HPLC

Product Introduction

Bioactivity
Description
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM).
Targets&IC50
PKA:2.3 nM(ki)
Chemical Properties
Molecular Weight2282.43
FormulaC96H152N32O33
SmilesCC[C@H](C)[C@@H](C(=O)N[C@@H](CC1=CNC=N1)C(=O)N[C@@H](CC(=O)O)C(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC3=CC=C(C=C3)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)N.CC(=O)O
Relative Density.1.31g/cm3
SequenceH-Thr-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-His-Asp-OH.CH3CO2H
Sequence ShortTTYADFIASGRTGRRNAIHD
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 2.5 mM, Sonication is recommended.
DMSO: Insoluble
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM0.4381 mL2.1906 mL4.3813 mL21.9065 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PKI (524) Acetate(99534039 free base)PKI (5 24) Acetate(99534 03 9 free base)PKI Acetate(99534-03-9 free base)PKA
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