Powder: -20°C for 3 years | In solvent: -80°C for 1 year
QCA570 is an effective BET degrader based on PROTAC (IC50: 10 nM for BRD4 BD1 Protein).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | Inquiry | |
50 mg | 10-14 weeks | Inquiry | |
100 mg | 10-14 weeks | Inquiry |
Description | QCA570 is an effective BET degrader based on PROTAC (IC50: 10 nM for BRD4 BD1 Protein). |
Targets&IC50 | BRD4 BD1:10 nM |
In vitro | QCA570 inhibits cell growth in MV4;11, MOLM-13, and RS4;11 cell lines (IC50: 8.3, 62, and 32 pM, respectively). QCA570 is an extremely effective and highly efficacious BET degrader, capable of degrading BET proteins at low picomolar (pM) concentrations in leukemia cells. [1]. |
Molecular Weight | 695.79 |
Formula | C39H33N7O4S |
CAS No. | 2207569-08-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
QCA570 2207569-08-0 Others QCA-570 QCA 570 inhibitor inhibit