Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 2,220.00 | |
50 mg | 10-14 weeks | $ 2,890.00 | |
100 mg | 10-14 weeks | $ 4,390.00 |
Description | CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM). |
Targets&IC50 | CCR2:2.4 nM (ki) |
In vitro | The combination of SAR and SKR in the hit-to-lead process results in the discovery of a new high-affinity and long residence time CCR2 antagonist 1 (compound 15a, Ki=2.4 nM; RT=714 min). |
Molecular Weight | 549.47 |
Formula | C28H32BrF3N2O |
CAS No. | 1683534-96-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
CCR2 antagonist 1 1683534-96-4 Immunology/Inflammation Microbiology/Virology CCR CCR-2 antagonist 1 inhibitor inhibit