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TargetMol | Compound Library

FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds. Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules. TargetMol's FDA-Approved & Pharmacopeia Drug Library collects 3270 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1010

FDA-Approved & Pharmacopeia Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • 3270 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
  • All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Autophagy
Endogenous Metabolite
Apoptosis
Adrenergic Receptor
5-HT Receptor
AChR
Parasite
COX
Histamine Receptor
Dopamine Receptor
Antifungal
HIV Protease
Sodium Channel
Calcium Channel
Potassium Channel
DNA/RNA Synthesis
NF-κB
Glucocorticoid Receptor
Estrogen/progestogen Receptor
Topoisomerase
Reactive Oxygen Species
Cytochromes P450
Influenza Virus
SARS-CoV
Ferroptosis
PDE
RAAS
GABA Receptor
EGFR
Dehydrogenase
Mitophagy
VEGFR
HCV Protease
Estrogen Receptor/ERR
PPAR
HSV
c-Kit
Microtubule Associated
Serotonin Transporter
Cholinesterase (ChE)
PDGFR
Nucleoside Antimetabolite/Analog
Prostaglandin Receptor
Reverse Transcriptase
ribosome
Antioxidant
MAO
Virus Protease
Progesterone Receptor
Norepinephrine
HBV
Proteasome
TRP/TRPV Channel
ATPase
iGluR
HDAC
Carbonic Anhydrase
FGFR
TNF
Antifection
JAK
MMP
Proton pump
Androgen Receptor
Monoamine Oxidase
Src
DNA Alkylator/Crosslinker
Bcr-Abl
ROS
Opioid Receptor
FLT
Transferase
Adenosine Receptor
Tyrosine Kinases
PKC
DPP-4
IL Receptor
Antiviral
Thrombin
HIF/HIF Prolyl-Hydroxylase
Phosphatase
c-Met/HGFR
MRP
NMDAR
Lipoxygenase
AMPK
HMG-CoA Reductase
Thyroid hormone receptor(THR)
PI3K
PARP
Drug Metabolite
GluR
STAT
NO Synthase
Antifolate
Raf
CDK
Mitochondrial Metabolism
Interleukin
ALK
Beta Amyloid
Retinoid Receptor
DHFR
Amino Acids and Derivatives
ERK
SGLT
P-gp
c-RET
Tyrosinase
DNA Alkylation
mTOR
Akt
HSP
TLR
Nrf2
Phospholipase
MEK
Factor Xa
Serine Protease
Endothelin Receptor
CaMK
Chloride channel
p38 MAPK
P2Y Receptor
ROCK
ABC Transporter
S1P Receptor
ADC Cytotoxin
Histone Methyltransferase
Integrin
Reductase
NADPH
PKA
Cysteine Protease
P2X Receptor
DNA gyrase
Monoamine Transporter
Trk receptor
Aromatase
HIF
DNA Methyltransferase
CFTR
HER
LPL Receptor
Glutathione Peroxidase
GNRH Receptor
Wnt/beta-catenin
FXR
Caspase
Guanylate cyclase
Hedgehog/Smoothened
Vasopressin Receptor
DNA
TGF-beta/Smad
PGE Synthase
Bcl-2 Family
IκB/IKK
GPR
Hydroxylase
Neurokinin receptor
Sigma receptor
TAM Receptor
ROS Kinase
NOS
GSK-3
Annexin A
Fatty Acid Synthase
Xanthine Oxidase
Cannabinoid Receptor
Anti-infection
FAK
Cell wall
Histone Demethylase
Melatonin Receptor
Serine/threonin kinase
Aryl Hydrocarbon Receptor
UGT
MT Receptor
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Smo
Lipid
GPCR19
Decarboxylase
Neprilysin
c-Fms
Ligand for E3 Ligase
CGRP Receptor
Gap Junction Protein
NOD
AhR
NOD-like Receptor (NLR)
MicroRNA
Arginase
CETP
JNK
CaSR
Cholecystokinin Receptor
Leukotriene Receptor
LDL
Gamma-secretase
Na-K-Cl cotransporter
Glucosidase
PAK
CCR
CXCR
Aurora Kinase
IGF-1R
OAT
Free radical scavengers
Aminopeptidase
Sirtuin
GluCls
GST
Oxytocin Receptor
Adenosine Deaminase
Complement System
Syk
Imidazoline Receptor
p53
Vitamin
BTK
Monocarboxylate transporter
ROR
CRM1
Ligands for Target Protein for PROTAC
YAP
LTR
IFNAR
TOPK
Rho
CSF-1R
Immunology/Inflammation related
IRE1
Adiponectin Receptor
GlyT
Hexokinase
Integrase
Thrombopoietin Receptor
Epigenetic Reader Domain
DUB
Indoleamine 2,3-Dioxygenase (IDO)
Telomerase
Beta-Secretase
Glutathione reductase
MAPK
Acyltransferase
Ephrin Receptor
RSV
Kras
Melanocortin Receptor
PDK
GHSR
PLK
Platelet aggregation
S6 Kinase
Ras
Protease-activated Receptor
PKM
Advanced Glycation End Products
Mdm2
Taste receptor
NPC1L1
Hydrogenase
RAR/RXR
DNA-PK
Dynamin
BACE
Na+/Ca2+ Exchanger
DYRK
Lipase
gp120/CD4
VDA
N-Acetylglucosaminyltransferase
Hck
Liver X Receptor
Glucokinase
RANKL/RANK
IAP
Myosin
PAFR
MTH1
GRK
Glucagon Receptor
Phosphorylase
Anion Exchanger
PROTAC Linker
HCN Channel
FAAH
ACK1
Angiotensin-converting Enzyme (ACE)
Somatostatin
Chk
PAD
Epoxide Hydrolase
cAMP
Mucin
ATP Citrate Lyase
STING
Histone Acetyltransferase
transporter
CRFR
Pyroptosis
Casein Kinase
CRISPR/Cas9
Aquaporin
NADPH-oxidase
IRAK
PD-1/PD-L1

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