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TargetMol | Compound Library

FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules.

TargetMol's FDA-Approved & Pharmacopeia Drug Library collects 3280 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1010

FDA-Approved & Pharmacopeia Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • 3280 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
  • All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Apoptosis
Endogenous Metabolite
Autophagy
Adrenergic Receptor
Parasite
5-HT Receptor
AChR
COX
Dopamine Receptor
Antifungal
Histamine Receptor
Potassium Channel
Calcium Channel
DNA/RNA Synthesis
Sodium Channel
HIV Protease
NF-κB
Reactive Oxygen Species
Cytochromes P450
SARS-CoV
Glucocorticoid Receptor
Virus Protease
Topoisomerase
Estrogen/progestogen Receptor
Influenza Virus
Ferroptosis
PDE
GABA Receptor
VEGFR
Estrogen Receptor/ERR
RAAS
Dehydrogenase
Mitophagy
EGFR
HCV Protease
HSV
Cholinesterase (ChE)
Serotonin Transporter
Microtubule Associated
c-Kit
PPAR
Nucleoside Antimetabolite/Analog
iGluR
TNF
PDGFR
Prostaglandin Receptor
Reverse Transcriptase
MMP
Interleukin
Progesterone Receptor
ribosome
HBV
Antioxidant
TRP/TRPV Channel
MAO
Norepinephrine
Proteasome
ATPase
HDAC
FGFR
Monoamine Oxidase
Carbonic Anhydrase
p38 MAPK
Drug Metabolite
Angiotensin-converting Enzyme (ACE)
Akt
Caspase
Antifection
JAK
PI3K
Opioid Receptor
Androgen Receptor
Proton pump
c-Met/HGFR
ERK
Bcl-2 Family
HIF/HIF Prolyl-Hydroxylase
DNA Alkylator/Crosslinker
Bcr-Abl
CDK
STAT
NO Synthase
ROS
FLT
Anti-infection
Transferase
Src
Adenosine Receptor
Tyrosine Kinases
Mitochondrial Metabolism
DPP-4
IL Receptor
Antiviral
Nrf2
AMPK
Amino Acids and Derivatives
Phosphatase
MRP
PARP
PKC
NMDAR
Beta Amyloid
HMG-CoA Reductase
Tyrosinase
Thrombin
Thyroid hormone receptor(THR)
Raf
Lipoxygenase
P-gp
HSP
GluR
ALK
Antifolate
mTOR
TLR
Phospholipase
MEK
Ras
DHFR
JNK
Serine Protease
SGLT
Retinoid Receptor
c-RET
DNA Alkylation
IκB/IKK
ROS Kinase
Factor Xa
Wnt/beta-catenin
Endothelin Receptor
CaMK
Sigma receptor
ADC Cytotoxin
Chloride channel
P2Y Receptor
PKA
ROCK
DNA gyrase
ABC Transporter
Monoamine Transporter
HIF
CFTR
S1P Receptor
Histone Methyltransferase
Integrin
LPL Receptor
Reductase
NADPH
Glutathione Peroxidase
GSK-3
FXR
P2X Receptor
TGF-beta/Smad
Trk receptor
Aromatase
Hydroxylase
MDM-2/p53
Neurokinin receptor
DNA Methyltransferase
HER
GPCR
GNRH Receptor
Cysteine Protease
Leukotriene Receptor
Glucosidase
Guanylate cyclase
Isocitrate Dehydrogenase (IDH)
Hedgehog/Smoothened
Vasopressin Receptor
Xanthine Oxidase
DNA
PGE Synthase
GPCR19
Kras
Complement System
TAM Receptor
NOD-like Receptor (NLR)
NOS
Melatonin Receptor
Serine/threonin kinase
Annexin A
Gamma-secretase
Molecular Glues
Fatty Acid Synthase
Aurora Kinase
IGF-1R
Telomerase
FAK
Cell wall
Histone Demethylase
CaSR
Aryl Hydrocarbon Receptor
UGT
MT Receptor
Na-K-Cl cotransporter
Smo
Thrombopoietin Receptor
Lipid
OAT
Aminopeptidase
Sirtuin
Decarboxylase
Neprilysin
FKBP
Ligand for E3 Ligase
c-Fms
Cannabinoid Receptor
Gap Junction Protein
NOD
AhR
Vitamin
MicroRNA
ASBT
Arginase
Cholecystokinin Receptor
Immunology/Inflammation related
LDL
BTK
Hexokinase
PAK
CCR
CXCR
Mucin
OXPHOS
MAPK
Free radical scavengers
GluCls
GST
Melanocortin Receptor
Oxytocin Receptor
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Syk
Imidazoline Receptor
p53
PD-1/PD-L1
IKZF
Monocarboxylate transporter
ROR
MTP
CRM1
Ligands for Target Protein for PROTAC
YAP
LTR
Na+/Ca2+ Exchanger
IFNAR
DYRK
Necroptosis
Tie-2
TOPK
Photosensitizer
Rho
NR4A
IDO
CSF-1R
Prolyl Endopeptidase (PREP)
IRE1
Adiponectin Receptor
PAFR
GlyT
Integrase
FAAH
PTEN
Epigenetic Reader Domain
DUB
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
Beta-Secretase
Glutathione reductase
Survivin
Acyltransferase
Ephrin Receptor
transporter
Pyroptosis
Casein Kinase
RSV
PDK
GHSR
PLK
Platelet aggregation
S6 Kinase
Protease-activated Receptor
PKM
Advanced Glycation End Products
Mdm2
Taste receptor
CAT
NPC1L1
Hydrogenase
DNA-PK
Dynamin
BACE
Lipase
CETP
gp120/CD4
MIF
VDA
OCT
c-Myc
N-Acetylglucosaminyltransferase
Hck
ATG
Liver X Receptor
Glucokinase
Glutaminase
RANKL/RANK
IAP
Myosin
E1/E2/E3 Enzyme
MTH1
GRK
Glucagon Receptor
Phosphorylase
Arp2/3 Complex
Anion Exchanger
PROTAC Linker
HCN Channel
Somatostatin
Chk
PAD
Epoxide Hydrolase
cAMP
BCRP
STING
Histone Acetyltransferase
CRFR
p62
TMV
CRISPR/Cas9
Aquaporin
NADPH-oxidase
IRAK

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