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TargetMol | Compound Library

FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds. Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules. TargetMol’s FDA-Approved & Pharmacopeia Drug Library collects 3158 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1010

FDA-Approved & Pharmacopeia Drug Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • 3158 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
  • All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Autophagy
Endogenous Metabolite
Apoptosis
Adrenergic Receptor
5-HT Receptor
AChR
COX
Parasite
Histamine Receptor
Dopamine Receptor
Antifungal
HIV Protease
Sodium Channel
Calcium Channel
DNA/RNA Synthesis
Potassium Channel
NF-κB
Topoisomerase
Reactive Oxygen Species
Estrogen/progestogen Receptor
Glucocorticoid Receptor
Influenza Virus
P450
Ferroptosis
PDE
SARS-CoV
RAAS
GABA Receptor
Dehydrogenase
Mitophagy
EGFR
HCV Protease
VEGFR
c-Kit
ribosome
HSV
PDGFR
PPAR
Serotonin Transporter
Nucleoside Antimetabolite/Analog
Prostaglandin Receptor
AChE
Microtubule Associated
Estrogen Receptor/ERR
Reverse Transcriptase
MAO
Virus Protease
Progesterone Receptor
Norepinephrine
HBV
Antioxidant
Proteasome
Antifection
iGluR
ATPase
FGFR
Carbonic Anhydrase
Androgen Receptor
TNF
JAK
HDAC
TRP/TRPV Channel
Monoamine Oxidase
Proton pump
MMP
FLT
Thrombin
Opioid Receptor
Adenosine Receptor
PKC
Src
DNA Alkylator/Crosslinker
Bcr-Abl
Transferase
ROS
IL Receptor
DPP-4
Antiviral
c-Met/HGFR
Tyrosine Kinases
Phosphatase
Drug Metabolite
MRP
GluR
NMDAR
HIF/HIF Prolyl-Hydroxylase
PI3K
Lipoxygenase
CDK
NO Synthase
Raf
AMPK
DHFR
Retinoid Receptor
HMG-CoA Reductase
ERK
GNRH Receptor
Tyrosinase
Thyroid hormone receptor(THR)
ALK
STAT
Interleukin
SGLT
P-gp
Amino Acids and Derivatives
PARP
Antifolate
Beta Amyloid
Phospholipase
mTOR
Mitochondrial Metabolism
Akt
Factor Xa
Nrf2
c-RET
MEK
HER
DNA Alkylation
DNA gyrase
BTK
CaMK
Serine Protease
ABC
Chloride channel
TLR
p38 MAPK
P2Y Receptor
CAT
TAM Receptor
Monoamine Transporter
DNA Methyltransferase
Cysteine Protease
Reductase
GPR
Neurokinin receptor
S1P Receptor
PKA
CFTR
NADPH
BCL
Trk receptor
Endothelin Receptor
LPL Receptor
HSP
P2X Receptor
Aromatase
ROCK
Glutathione Peroxidase
Caspase
Hedgehog/Smoothened
Histone Methyltransferase
IκB/IKK
Wnt/beta-catenin
TGF-beta/Smad
Cannabinoid Receptor
HIF
Vasopressin Receptor
Annexin A
ROS Kinase
Anti-infection
DNA
Xanthine Oxidase
FXR
Hydroxylase
Lipid
PGE Synthase
Cell wall
Serine/threonin kinase
GSK-3
Integrin
Ras
FAK
Fatty Acid Synthase
Guanylate cyclase
Histone Demethylase
NOS
MT Receptor
Decarboxylase
Neprilysin
GPCR19
NOD-like Receptor (NLR)
Gamma-secretase
CaSR
Melatonin Receptor
Smo
AhR
NOD
Sigma receptor
UGT
Aryl Hydrocarbon Receptor
Oxytocin Receptor
p53
c-Fms
Leukotriene Receptor
PKM
LDL
CXCR
Hexokinase
Ligand for E3 Ligase
Adenosine deaminase
Free radical scavengers
cholecystokinin
Aminopeptidase
CETP
JNK
Glucosidase
Sirtuin
Syk
Imidazoline Receptor
GST
Arginase
IGF-1R
Molecular Glues
Isocitrate Dehydrogenase (IDH)
CCR
Na-K-Cl cotransporter
GluCls
Aurora Kinase
Gap Junction Protein
PAK
Melanocortin Receptor
S6 Kinase
DUB
PLK
Somatostatin
IRE1
RSV
CRM1
YAP
PDK
ROR
MAPK
Platelet aggregation
TOPK
Monocarboxylate transporter
OAT
Adiponectin receptor
Rho
Glutathione reductase
Telomerase
DYRK
Ligands for Target Protein for PROTAC
Immunology/Inflammation related
Complement System
Protease-activated Receptor
Ephrin Receptor
LTR
GlyT
Integrase
Indoleamine 2,3-Dioxygenase (IDO)
Beta-Secretase
Thrombopoietin Receptor
IFNAR
Acyltransferase
CGRP Receptor
Phosphorylase
Epigenetic Reader Domain
NADPH-oxidase
RAR/RXR 
Casein Kinase
Lipase
Pyroptosis
IAP
Mdm2
MTH1
GHSR
Aquaporin
transporter
Anion Exchanger
NPC1L1
Bradykinin Receptor
GRK
Glucokinase
CSF-1R
CRISPR/Cas9
advanced glycation end products
PAFR
Taste receptor
Liver X Receptor
Epoxide Hydrolase
FAAH
Hydrogenase
RANKL/RANK
Histone Acetyltransferase
VDA
PROTAC Linker
N-Acetylglucosaminyltransferase
Dynamin
Glucagon Receptor
gp120/CD4
cAMP
BACE
Na+/Ca2+ Exchanger
DNA-PK
STING
OX Receptor
ACK
PD-1/PD-L1
Myosin
PAD
Chk
Angiotensin-converting Enzyme (ACE)
Hck
IRAK
ATP Citrate Lyase

Keywords