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RG-102240 (Synonyms: RG102240, RG 102240)

Name: RG-102240
Brand: TargetMol
SKU: T28530
Price: 76 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T28530 Copy Product Info

Purity: 99.81%

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RG-102240 is a ligand for the insect ecdysone receptor (EcR). Its IC50 values against wild-type G:CfE (DEF) and A110P mutant are 85 nM and 13 nM, respectively. It activates reporter gene expression of both wild-type CfEcR and the A110P mutant.

RG-102240

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Catalog No. T28530

Synonyms RG102240, RG 102240

Cas No. 162326-49-0

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Pack Size	Price	USA Stock	Global Stock
1 mg	$76	-	In Stock
5 mg	$185	-	In Stock
10 mg	$297	-	In Stock
25 mg	$596	-	In Stock
50 mg	$953	-	In Stock
100 mg	$1,520	-	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:99.81%

Appearance:Solid

Color:White

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COA LCMS HNMR

Product Introduction

Bioactivity

Description	RG-102240 is a ligand for the insect ecdysone receptor (EcR). Its IC50 values against wild-type G:CfE (DEF) and A110P mutant are 85 nM and 13 nM, respectively. It activates reporter gene expression of both wild-type CfEcR and the A110P mutant.
Targets&IC50	A110P mutant:13 nM, Wild type G:CfE (DEF):85 nM
Synonyms	RG102240, RG 102240

Chemical Properties

Molecular Weight	382.5
Formula	C₂₃H₃₀N₂O₃
Cas No.	162326-49-0
Smiles	O=C(NN(C(=O)C=1C=C(C=C(C1)C)C)C(C)(C)C)C=2C=CC=C(OC)C2CC
Relative Density.	1.086 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (209.15 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.6144 mL	13.0719 mL	26.1438 mL	130.7190 mL
5 mM	0.5229 mL	2.6144 mL	5.2288 mL	26.1438 mL
10 mM	0.2614 mL	1.3072 mL	2.6144 mL	13.0719 mL
20 mM	0.1307 mL	0.6536 mL	1.3072 mL	6.5359 mL
50 mM	0.0523 mL	0.2614 mL	0.5229 mL	2.6144 mL
100 mM	0.0261 mL	0.1307 mL	0.2614 mL	1.3072 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc