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CP-8668

Catalog No. T31082 CAS 209331-43-1

Synonyms: UNII-5371O2R79D, CP 8668

CP-8668 is an orally active nonsteroidal progesterone receptor modulator with tetrahydrobenzoindolone skeleton.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

CP-8668, CAS 209331-43-1

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25 mg	Inquiry	$ 1,520.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

CP-8668 is an orally active nonsteroidal progesterone receptor modulator with tetrahydrobenzoindolone skeleton.

Synonyms	UNII-5371O2R79D, CP 8668
Molecular Weight	374.47
Formula	C21H30N2O4
CAS No.	209331-43-1

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Kurihara K, Shinei R, Tanabe K, Tabata Y, Kurata Y, Hoshiko S, Okonogi T. Nonsteroidal progesterone receptor ligands (II); synthesis and SAR of new tetrahydrobenzindolone derivatives. Bioorg Med Chem. 2006 Jul 15;14(14):4862-78. Epub 2006 Mar 31. PubMed PMID: 16580209. 2. Tabata Y, Iizuka Y, Shinei R, Kurihara K, Okonogi T, Hoshiko S, Kurata Y. CP8668, a novel orally active nonsteroidal progesterone receptor modulator with tetrahydrobenzindolone skeleton. Eur J Pharmacol. 2003 Feb 7;461(1):73-8. Erratum in: Eur J Pharmacol. 2003 Apr 4;465(3):299. PubMed PMID: 12568918.

Dose Conversion

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Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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The answer of 19.713 mg appears in the Mass box

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An example of a dilution calculation using the Tocris dilution calculator
What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
Using the equation C1V1 = C2V2, where C1=10 mM, C2=50 μM, V2=20 ml and V1 is the unknown:
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The answer of 100 microliter (0.1 ml) appears in the Volume (start) box

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

CP-8668 209331-43-1 UNII-5371O2R79D CP8668 CP 8668 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.