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Scyliorhinin I

Name: Scyliorhinin I
Brand: TargetMol
SKU: TP2785
Rating: 4.5 (1 reviews)

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Catalog No. TP2785Cas No. 103425-21-4

Scyliorhinin I is an agonist for both neurokinin-1 (NK-1) and neurokinin-2 (NK-2) receptors, exhibiting a Ki value of 0.9 nM at rat submandibular gland NK-1 receptors and 2 nM at hamster bladder NK-2 receptors. Additionally, it possesses the capability to contract the longitudinal muscle of the guinea pig ileum.

Scyliorhinin I

😃Good

Catalog No. TP2785Cas No. 103425-21-4

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
10 mg	Inquiry	Inquiry	Inquiry
50 mg	Inquiry	Inquiry	Inquiry

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Product Introduction

Bioactivity

Description	Scyliorhinin I is an agonist for both neurokinin-1 (NK-1) and neurokinin-2 (NK-2) receptors, exhibiting a Ki value of 0.9 nM at rat submandibular gland NK-1 receptors and 2 nM at hamster bladder NK-2 receptors. Additionally, it possesses the capability to contract the longitudinal muscle of the guinea pig ileum.
Targets&IC50	NK-2 (guinea pig):2 nM (Ki), NK1 (rat):0.9 nM (Ki)

Chemical Properties

Molecular Weight	1218.47
Formula	C₅₉H₈₇N₁₃O₁₃S
Cas No.	103425-21-4
Smiles	[C@H](CC1=CC=CC=C1)(C(N[C@@H](CC2=CC=C(O)C=C2)C(NCC(N[C@H](C(N[C@@H](CCSC)C(N)=O)=O)CC(C)C)=O)=O)=O)NC([C@@H](NC([C@@H](NC([C@H](CC3=CC=CC=C3)NC([C@H](CCCCN)NC([C@H](C)N)=O)=O)=O)CC(O)=O)=O)CCCCN)=O

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline /PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline /PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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