Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Anti-Cancer Approved Drug Library

Catalog No. L2110

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 1800 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L2110

Anti-Cancer Approved Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 1800 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Sci Citations

Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
5-HT Receptor
Adrenergic Receptor
Endogenous Metabolite
Antibacterial
COX
Antibiotic
Dopamine Receptor
Histamine Receptor
Sodium Channel
Potassium Channel
DNA/RNA Synthesis
Calcium Channel
AChR
Parasite
Glucocorticoid Receptor
HIV Protease
Cytochromes P450
EGFR
Estrogen/progestogen Receptor
NF-κB
VEGFR
Antifungal
GABA Receptor
Reactive Oxygen Species
Ferroptosis
Topoisomerase
c-Kit
Mitophagy
PDGFR
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
PPAR
SARS-CoV
Dehydrogenase
Microtubule Associated
PDE
Prostaglandin Receptor
Influenza Virus
Serotonin Transporter
ATPase
HDAC
iGluR
Norepinephrine
FGFR
JAK
Androgen Receptor
HSV
Proton pump
Bcr-Abl
DNA Alkylator/Crosslinker
FLT
RAAS
Src
Adenosine Receptor
c-Met/HGFR
TRP/TRPV Channel
Tyrosine Kinases
HBV
Opioid Receptor
Virus Protease
Progesterone Receptor
TNF
ALK
NMDAR
PKC
Raf
ROS
CDK
HMG-CoA Reductase
PARP
Retinoid Receptor
SGLT
AMPK
Antifolate
Carbonic Anhydrase
Cholinesterase (ChE)
c-RET
DHFR
Drug Metabolite
GNRH Receptor
MAO
MMP
MRP
P-gp
Phosphatase
Reverse Transcriptase
DNA Alkylation
HCV Protease
Lipoxygenase
PI3K
Proteasome
ABC Transporter
Antifection
CaMK
GluR
HIF/HIF Prolyl-Hydroxylase
Interleukin
P2Y Receptor
STAT
ADC Cytotoxin
CFTR
Chloride channel
DNA Methyltransferase
Guanylate cyclase
HER
IL Receptor
MEK
Monoamine Oxidase
NADPH
Phospholipase
S1P Receptor
Thrombin
TLR
Trk receptor
Aromatase
Endothelin Receptor
FXR
Hedgehog/Smoothened
Histone Methyltransferase
HSP
Mitochondrial Metabolism
Monoamine Transporter
Neurokinin receptor
Nrf2
P2X Receptor
PKA
ROCK
ROS Kinase
TAM Receptor
Transferase
Bcl-2 Family
Beta Amyloid
Caspase
DNA
Glutathione Peroxidase
GPCR
HIF
LPL Receptor
mTOR
ribosome
Sigma receptor
Vasopressin Receptor
Akt
Amino Acids and Derivatives
Annexin A
Antioxidant
Antiviral
CaSR
DPP-4
ERK
Fatty Acid Synthase
GPCR19
GSK-3
Isocitrate Dehydrogenase (IDH)
IκB/IKK
Ligand for E3 Ligase
Melatonin Receptor
Molecular Glues
NO Synthase
NOD
Oxytocin Receptor
PGE Synthase
Smo
Tyrosinase
Wnt/beta-catenin
Xanthine Oxidase
Adenosine Deaminase
AhR
Aminopeptidase
c-Fms
Cysteine Protease
Decarboxylase
FAK
Free radical scavengers
Gamma-secretase
Hydroxylase
IGF-1R
Integrin
Leukotriene Receptor
Melanocortin Receptor
MicroRNA
MT Receptor
Na-K-Cl cotransporter
p38 MAPK
PAK
Serine Protease
Serine/threonin kinase
Syk
TGF-beta/Smad
UGT
BTK
Arginase
Aryl Hydrocarbon Receptor
Aurora Kinase
Beta-Secretase
Cannabinoid Receptor
CCR
Cell wall
CGRP Receptor
Cholecystokinin Receptor
CRM1
CXCR
DNA gyrase
Ephrin Receptor
Gap Junction Protein
GHSR
GST
Hexokinase
IFNAR
IRE1
Kras
LDL
Ligands for Target Protein for PROTAC
LTR
MAPK
Monocarboxylate transporter
NOD-like Receptor (NLR)
NOS
OAT
PLK
Protease-activated Receptor
Ras
Reductase
Rho
ROR
RSV
YAP
ACK1
Adiponectin Receptor
ATP Citrate Lyase
BACE
Bradykinin Receptor
cAMP
Chk
Complement System
CSF-1R
DNA-PK
DUB
Epigenetic Reader Domain
FAAH
Factor Xa
Glucagon Receptor
GluCls
Glutathione reductase
gp120/CD4
GRK
Hck
HCN Channel
Histone Demethylase
Hydrogenase
IAP
Imidazoline Receptor
Immunology/Inflammation related
Indoleamine 2,3-Dioxygenase (IDO)
Lipase
Lipid
Liver X Receptor
Mdm2
MTH1
Na+/Ca2+ Exchanger
NADPH-oxidase
Neprilysin
NPC1L1
p53
PAD
PAFR
PD-1/PD-L1
PDK
Platelet aggregation
PROTAC Linker
Pyroptosis
S6 Kinase
Sirtuin
Somatostatin
STING
Thrombopoietin Receptor
TOPK
VDA

Keywords