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Zaurategrast ethyl ester sulfate

Catalog No. T13388 CAS 1214261-78-5

Synonyms: UCB1184197 sulfate, CDP323 sulfate

Zaurategrast ethyl ester sulfate is a α4β1/α4β7 integrin antagonist, and used for the treatment of inflammatory and autoimmune disorders.

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Zaurategrast ethyl ester sulfate Chemical Structure

Zaurategrast ethyl ester sulfate, CAS 1214261-78-5

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,670.00
50 mg	6-8 weeks	$ 2,180.00
100 mg	6-8 weeks	$ 2,800.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Zaurategrast ethyl ester sulfate is a α4β1/α4β7 integrin antagonist, and used for the treatment of inflammatory and autoimmune disorders.
In vitro	Zaurategrast ethyl ester sulfate is an ethyl ester prodrug of CT7758, shows some improvements in increasing mass transfer[1].

Synonyms	UCB1184197 sulfate, CDP323 sulfate
Molecular Weight	1197.01
Formula	C56H60Br2N8O10S
CAS No.	1214261-78-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Chanteux H, et al. Cross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin Antagonist. Drug Metab Dispos. 2015 Sep;43(9):1381-91. 2. Davenport RJ, et al. Alpha4-integrin antagonism--an effective approach for the treatment of inflammatory diseases? Drug Discov Today. 2007 Jul;12(13-14):569-76.

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Keywords

Zaurategrast ethyl ester sulfate 1214261-78-5 Others UCB1184197 sulfate CDP323 sulfate CDP 323 Sulfate CDP323 Sulfate UCB1184197 Sulfate CDP-323 Sulfate UCB 1184197 Sulfate Zaurategrast ethyl ester Sulfate UCB-1184197 Sulfate inhibitor inhibit

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