keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
YAP-TEAD-IN-1 TFA is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TEAD1 (Kd: 15 nM) than YAP (50-171) (Kd: 40 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | 5 days | $ 150.00 | |
5 mg | 5 days | $ 344.00 | |
10 mg | 5 days | $ 571.00 |
Description | YAP-TEAD-IN-1 TFA is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TEAD1 (Kd: 15 nM) than YAP (50-171) (Kd: 40 nM). |
Targets&IC50 | YAP-TEAD:25 nM |
In vitro | In a GST pull-down assay, YAP-TEAD-IN-1 (2 μM) is against endogenous YAP binding to GST-TEAD (1209-426), the Kd of His-YAP1209-426 is determined to be 40 nM. |
Molecular Weight | N/A |
Formula | C93H144ClN23O21S2.xC2HF3O2 |
CAS No. | 1659305-79-9 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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YAP-TEAD-IN-1 TFA 1659305-79-9 Others YAPTEADIN1 TFA YAP TEAD IN 1 TFA inhibitor inhibit