Powder: -20°C for 3 years | In solvent: -80°C for 1 year
OMDM169 is a potent and selective MAGL inhibitor. OMDM169 could enhances 2-AG levels and of exerts analgesic activity via indirect activation of cannabinoid receptors. OMDM169 exhibited 0.13 microM<IC(50)<0.41 microM towards 2-AG hydrolysing activities in rat cerebellum and COS-7 cells, and inhibited the human recombinant MAGL (IC(50)=0.89 microM), whilst being inactive at human CB(1) and CB(2) receptors (K(i)<10 microM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 2,720.00 | |
50 mg | 10-14 weeks | $ 3,580.00 | |
100 mg | 10-14 weeks | $ 4,900.00 |
Description | OMDM169 is a potent and selective MAGL inhibitor. OMDM169 could enhances 2-AG levels and of exerts analgesic activity via indirect activation of cannabinoid receptors. OMDM169 exhibited 0.13 microM<IC(50)<0.41 microM towards 2-AG hydrolysing activities in rat cerebellum and COS-7 cells, and inhibited the human recombinant MAGL (IC(50)=0.89 microM), whilst being inactive at human CB(1) and CB(2) receptors (K(i)>10 microM). |
Synonyms | OMDM 169, OMDM-169 |
Molecular Weight | 439.63 |
Formula | C25H45NO5 |
CAS No. | 130193-44-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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OMDM169 130193-44-1 OMDM 169 OMDM-169 inhibitor inhibit