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CPI-169

Catalog No. T27069   CAS 1802175-07-0
Synonyms: CPI 169 (R), CPI-169 (R)

CPI-169 (R) is a novel and potent inhibitor of EZH2.

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CPI-169 Chemical Structure
CPI-169, CAS 1802175-07-0
Pack Size Availability Price/USD Quantity
25 mg 8-10 weeks $ 1,970.00
50 mg 8-10 weeks $ 2,580.00
100 mg 8-10 weeks $ 3,400.00
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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.
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Biological Description
Chemical Properties
Storage & Solubility Information
Description CPI-169 (R) is a novel and potent inhibitor of EZH2.
Targets&IC50 EZH2 Y641N:0.51 nM (IC50), EZH2 WT:0.24 nM (IC50), EZH1:6.1 nM (IC50)
Synonyms CPI 169 (R), CPI-169 (R)
Molecular Weight 528.66
Formula C27H36N4O5S
CAS No. 1802175-07-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

TargetMolReferences and Literature

1. Jenoh EM, Robert EM, Lehmann I, Kioko E, Bosire JO, Ngisiange N, Dahdouh-Guebas F, Koedam N. Wide Ranging Insect Infestation of the Pioneer Mangrove Sonneratia alba by Two Insect Species along the Kenyan Coast. PLoS One. 2016 May 12;11(5):e0154849. doi: 10.1371/journal.pone.0154849. eCollection 2016. PubMed PMID: 27171470; PubMed Central PMCID: PMC4865246. 2. Murphy S, Dalton M, Dawes D. Assessing Physical Therapy Students' Performance during Clinical Practice. Physiother Can. 2014 Spring;66(2):169-76. doi: 10.3138/ptc.2013-26. PubMed PMID: 24799754; PubMed Central PMCID: PMC4006410. 3. Seng P, Abat C, Rolain JM, Colson P, Lagier JC, Gouriet F, Fournier PE, Drancourt M, La Scola B, Raoult D. Identification of rare pathogenic bacteria in a clinical microbiology laboratory: impact of matrix-assisted laser desorption ionization-time of flight mass spectrometry. J Clin Microbiol. 2013 Jul;51(7):2182-94. doi: 10.1128/JCM.00492-13. Epub 2013 May 1. PubMed PMID: 23637301; PubMed Central PMCID: PMC3697718. 4. Nfotabong-Atheull A, Din N, Essomè Koum LG, Satyanarayana B, Koedam N, Dahdouh-Guebas F. Assessing forest products usage and local residents' perception of environmental changes in peri-urban and rural mangroves of Cameroon, Central Africa. J Ethnobiol Ethnomed. 2011 Dec 6;7:41. doi: 10.1186/1746-4269-7-41. PubMed PMID: 22146073; PubMed Central PMCID: PMC3261808.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

CPI-169 1802175-07-0 CPI 169 (R) CPI169 CPI-169 (R) CPI 169 inhibitor inhibit

 

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