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TargetMol | Compound Library

NMPA-Approved Drug Library

Catalog No. L4210

The NMPA Marketed Drug Library compiles 1580 compounds approved by the National Medical Products Administration (NMPA) of China. All compounds in this library have undergone clinical validation, possess well-defined targets, and demonstrate favorable safety profiles and bioavailability. This collection serves as an ideal resource for drug repurposing, significantly enhancing the success rate of drug development while shortening development timelines and reducing R&D costs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4210

NMPA-Approved Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1580 NMPA-approved drugs, ideal for high-throughput screening (HTS) and high-content screening (HCS).
  • All compounds are officially approved by the NMPA and accompanied by their corresponding NMPA approval numbers, making this library a powerful tool for drug repurposing and novel target identification.
  • Each compound has undergone rigorous preclinical studies and clinical trials, ensuring well-established biological activity and safety.
  • Spans multiple therapeutic areas, including oncology, cardiovascular diseases, anti-inflammatory agents, immunomodulators, central nervous system (CNS) drugs, respiratory therapeutics, and more.
  • Features structurally diverse compounds with potent pharmacological activity and excellent cell permeability.
  • Comprehensive documentation provided for each compound, including chemical structure, target information, IC₅₀ values, and detailed activity descriptions.
  • Compound identity and high purity are verified using multiple analytical techniques—including NMR、HPLC/LCMS—minimizing the risk of false positives.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Antibacterial
Antibiotic
Apoptosis
Autophagy
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
COX
DNA/RNA Synthesis
Parasite
Dopamine Receptor
Histamine Receptor
Calcium Channel
ROS
Potassium Channel
Antifungal
NF-κB
Sodium Channel
HIV Protease
Topoisomerase
Glucocorticoid Receptor
Cytochromes P450
Reactive Oxygen Species
Ferroptosis
Estrogen/progestogen Receptor
SARS-CoV
RAAS
Virus Protease
Nucleoside Antimetabolite/Analog
Akt
Interleukin
Influenza Virus
GABA Receptor
Serotonin Transporter
ERK
EGFR
Mitophagy
PDE
HSV
HBV
VEGFR
Prostaglandin Receptor
TNF
PPAR
Caspase
p38 MAPK
Microtubule Associated
Estrogen Receptor/ERR
iGluR
PDGFR
Reverse Transcriptase
Dehydrogenase
ribosome
Antifection
Opioid Receptor
c-Kit
Cholinesterase (ChE)
Proteasome
DNA Alkylator/Crosslinker
Angiotensin-converting Enzyme (ACE)
MMP
Norepinephrine
TLR
HCV Protease
JNK
Progesterone Receptor
TRP/TRPV Channel
Androgen Receptor
Bcl-2 Family
STAT
AMPK
HMG-CoA Reductase
ATPase
FGFR
NO Synthase
Proton pump
Amino Acids and Derivatives
Bcr-Abl
IL Receptor
mTOR
MRP
Wnt/beta-catenin
Thyroid hormone receptor(THR)
Carbonic Anhydrase
c-Met/HGFR
Adenosine Receptor
Drug Metabolite
Mitochondrial Metabolism
Phospholipase
Thrombin
HIF/HIF Prolyl-Hydroxylase
ADC Cytotoxin
Phosphatase
MAO
P-gp
Anti-infection
Antioxidant
Glutathione Peroxidase
Factor Xa
Raf
CDK
NMDAR
DPP-4
DNA Alkylation
CaMK
Beta Amyloid
MEK
Transferase
DHFR
Src
PI3K
GSK-3
Antifolate
PKC
Antiviral
HSP
Nrf2
ALK
HDAC
c-RET
FLT
Sigma receptor
Monoamine Oxidase
PKA
Leukotriene Receptor
FXR
Glucosidase
GluR
glycosidase
Retinoid Receptor
HIF
DNA Methyltransferase
Ras
Histone Methyltransferase
P2Y Receptor
Reductase
Necroptosis
PARP
Serine Protease
P2X Receptor
DNA gyrase
ABC Transporter
Na-K-Cl cotransporter
Fatty Acid Synthase
Vasopressin Receptor
Xanthine Oxidase
Lipoxygenase
SGLT
IκB/IKK
Aromatase
ROS Kinase
GPCR
NOS
Melatonin Receptor
GNRH Receptor
Tyrosine Kinases
Serine/threonin kinase
Cysteine Protease
ROCK
RANKL/RANK
IRE1
Annexin A
Molecular Glues
Endothelin Receptor
TGF-beta/Smad
PGE Synthase
Trk receptor
Free radical scavengers
Aminopeptidase
GPCR19
FKBP
Ligand for E3 Ligase
Complement System
MDM-2/p53
Tyrosinase
AhR
NOD-like Receptor (NLR)
Imidazoline Receptor
HER
Vitamin
IKZF
MicroRNA
Integrin
Arginase
LTR
Cell wall
NADPH
Lipase
PERK
Tie-2
TOPK
CaSR
Cholecystokinin Receptor
Rho
ATG
NR4A
UGT
PAFR
LDL
Gamma-secretase
MT Receptor
Hedgehog/Smoothened
JAK
Aurora Kinase
DNA
Mucin
Telomerase
MAPK
Neprilysin
GST
Kras
Oxytocin Receptor
Adenosine Deaminase
Gap Junction Protein
NOD
IRAK
CFTR
Advanced Glycation End Products
Mdm2
Chloride channel
NPC1L1
Monocarboxylate transporter
Hydrogenase
RAR/RXR
ROR
CRM1
Ligands for Target Protein for PROTAC
LPL Receptor
BACE
Na+/Ca2+ Exchanger
IFNAR
MIF
OCT
c-Myc
LDLR
Amylase
Aryl Hydrocarbon Receptor
IDO
E1/E2/E3 Enzyme
RIP kinase
GRK
Glucagon Receptor
Phosphorylase
Arp2/3 Complex
BTK
Monoamine Transporter
Guanylate cyclase
Smo
Integrase
PROTAC Linker
HCN Channel
PAK
FAAH
CCR
HCAR
PTEN
Somatostatin
Epoxide Hydrolase
Thrombopoietin Receptor
Epigenetic Reader Domain
IGF-1R
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
BCRP
Huntingtin
Glutathione reductase
Survivin
Acyltransferase
Sirtuin
Ephrin Receptor
transporter
Decarboxylase
ASK
RSV
ATM/ATR
p62
Melanocortin Receptor
CRISPR/Cas9
Aquaporin
Hydroxylase
FOXO
Cuproptosis
Cannabinoid Receptor
Neurokinin receptor
NADPH-oxidase
S6 Kinase
TAM Receptor
PD-1/PD-L1
S1P Receptor
Ferroportin

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