T78127 |
Tisolagiline
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1894207-44-3
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98%
|
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Tisolagiline (KDS2010), a reversible MAO-B inhibitor, is utilized in Parkinson's disease research [1].
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T78648 |
MAO-B-IN-3
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|
98%
|
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MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki o...
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T78649 |
MAO-B-IN-4
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98%
|
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MAO-B-IN-4 (Compound 26) is a reversible monoamine oxidase B (MAO-B) inhibitor with potent in vitro activity, characterized by an IC50 value of 9 nM. This orally...
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T78690 |
MAO-B-IN-18
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|
98%
|
|
MAO-B-IN-18 is a potent, selective inhibitor of MAO B, demonstrating IC50 values of 52 nM for hMAO B and 14 μM for hMAO A. It exhibits cytoprotective effects aga...
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T78793 |
MAOA-IN-1
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|
98%
|
|
MAOA-IN-1 (compound 15) is an orally-active inhibitor of monoamine oxidase A (MAOA) that exhibits cytotoxic effects on prostate cancer cells. This compound demon...
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T78821 |
IHC3
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98%
|
|
IHC3 is a competitive and reversible monoamine oxidase B (MAO-B) inhibitor with an IC50 of 1.672 μM, which targets Cys172 within the enzyme's active site. It is ...
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T78848 |
MAO-IN-3
|
797805-26-6
|
98%
|
|
MAO-IN-3 (Compound 5), a reversible and competitive monoamine oxidase (MAO) inhibitor with inhibition constants (K i) of 0.6 μM for MAO A and 0.2 μM for MAO B, e...
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T78859 |
MAO-B-IN-23
|
2107978-22-1
|
98%
|
|
MAO-B-IN-23, also known as Compound 11f, is a reversible and competitive monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 1.44 μM and a Ki of 0.51 μM ...
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T78860 |
MAO-B-IN-24
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|
98%
|
|
MAO-B-IN-24 (compound 11h) is a selective, reversible, competitive inhibitor of MAO-B with an IC50 value of 1.60 μM. It also exhibits inhibitory effects on MAO-A...
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T78889 |
Lysyl hydroxylase 2-IN-1
|
|
98%
|
|
"Lysyl Hydroxylase 2-IN-1 (compound 12) is a selective inhibitor of lysyl hydroxylase 2 (LH2) with an IC50 of approximately 300 nM and demonstrates specificity f...
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T78898 |
Lysyl hydroxylase 2-IN-2
|
|
98%
|
|
Lysyl Hydroxylase 2-IN-2 (compound 13) is a potent inhibitor of Lysyl Hydroxylase 2 (LH2), exhibiting an IC50 of approximately 500 nM. It effectively inhibits ce...
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T78907 |
MAO-B-IN-22
|
2902600-76-2
|
98%
|
|
MAO-B-IN-22 (compound 6h) represents a powerful MAO-B inhibitor, boasting an IC50 value of 0.014 μM, and exhibits high antioxidant activity alongside effective m...
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T79229 |
ETAP
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2575731-47-2
|
98%
|
|
ETAP, a dual inhibitor of both monoamine oxidase A (MAO-A) and monoamine oxidase B (MAO-B), exhibits antidepressant-like effects and is utilized in the research ...
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T79299 |
HAChE-IN-3
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|
98%
|
|
hAChE-IN-3 (compound 5c) serves as a potent inhibitor for AChE, BuChE, MAO-B, and BACE-1, with respective IC50 values of 0.44, 0.08, 5.15, and 0.38 μM, demonstra...
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T79486 |
MAO A/HSP90-IN-1
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2927489-95-8
|
98%
|
|
MAO A/HSP90-IN-1 (4-b) is a dual inhibitor of MAO A and HSP90, exhibiting IC50 values of 1.77 μM in glioblastoma (GBM) GL26 cells and 0.019 μM against HSP90α. Th...
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T79487 |
MAO A/HSP90-IN-2
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2927489-99-2
|
98%
|
|
MAO A/HSP90-IN-2 (compound 4-C), a dual inhibitor of HSP90 and MAO A, exhibits IC50 values of 0.016 μM for MAO A and 4.58 μM for HSP90. This compound not only en...
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T79761 |
MAO-B-IN-25
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|
98%
|
|
MAO-B-IN-25 (compound 92) is a selective inhibitor of monoamine oxidase B (MAO-B), exhibiting inhibitory half-maximal inhibitory concentrations (IC50) of 240 nM ...
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T79914 |
Tranylcypromine
|
155-09-9
|
98%
|
|
Tranylcypromine (SKF 385), a potent monoamine oxidase (MAO) inhibitor [1], is used in medicinal applications.
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T79979 |
Methyl piperate
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6190-46-1
|
98%
|
|
Methylpiperic acid, a piperine alkaloid, exhibits potent inhibitory activity on monoamine oxidase (MAO), with differing efficacy on isoforms: greater inhibition ...
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T80634 |
MAO-B-IN-19
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152897-41-1
|
98%
|
|
MAO-B-IN-19, a selective MAO-B inhibitor, exhibits neuroprotective and anti-inflammatory properties and demonstrates an IC50 value of 0.67 μM [1].
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