Home Tools
Log in
Products Inhibitors Libraries Recombinant Proteins Kits Services Contact Us
Cart
Peptides Monoclonal Antibodies Dye Reagents PROTAC Virtual Screening TargetMol Kits Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails Natural Products Phenols Alkaloids Flavonoids
Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK
Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library
TargetMol
Cytokines and Growth Factors •   Cytokines •   Growth Factors Receptor Proteins •   Fc Receptors •   Cytokines and Growth Factor Receptors
CD Proteins •   T Cell CD Proteins •   B Cell CD Proteins Immune Checkpoint Proteins •   Co-inhibitory Immune Checkpoint Proteins •   Co-stimulatory Immune Checkpoint Proteins
CAR-T Therapy Target Proteins •   Hematologic Malignancies Target Proteins •   Solid Tumors Target Proteins Enzymes •   Oxidoreductases,EC 1 •   Transferases,EC 2
Viral Proteins •   Coronavirus (CoV) Proteins •   Influenza Proteins Fluorescent Proteins Others

Anti-Cancer Approved Drug Library

Catalog No. L2110
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1779 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 1779 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (2.39 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2110)

Publications Cited TargetMol Libraries

1. Oncogene. 2021: 1-13.. 2. Cell Death & Disease. 2023, 14(4): 272. 3. British Journal of Cancer. 2023: 1-12. 4. Molecular oncology. 2022, 16(5): 1091. 5. Oncology Reports. 2023, 50(6): 1-11. 6. bioRxiv. 2023: 2023.01. 16.523559. 7. Cell Stem Cell. 2022 Apr 29(4) 545–558. 8. Science Bulletin. 2022. 9. Science Translational Medicine. 2022, 14(656): eabn3231.
Hide

Library Composition

Autophagy (332)
Apoptosis (245)
Adrenergic Receptor (157)
5-HT Receptor (156)
Endogenous Metabolite (140)
Antibacterial (133)
COX (118)
Antibiotic (111)
Dopamine Receptor (104)
Histamine Receptor (103)
Sodium Channel (77)
DNA/RNA Synthesis (76)
Potassium Channel (72)
Calcium Channel (71)
AChR (67)
Parasite (53)
Glucocorticoid Receptor (51)
P450 (43)
HIV Protease (42)
NF-κB (36)
Antifungal (36)
Reactive Oxygen Species (35)
Ferroptosis (33)
EGFR (33)
Estrogen/progestogen Receptor (33)
GABA Receptor (32)
VEGFR (32)
c-Kit (32)
Mitophagy (31)
Nucleoside Antimetabolite/Analog (29)
PPAR (29)
Topoisomerase (29)
PDGFR (29)
SARS-CoV (28)
Estrogen Receptor/ERR (27)
Dehydrogenase (27)
Influenza Virus (26)
Prostaglandin Receptor (26)
PDE (25)
Microtubule Associated (23)
Serotonin Transporter (23)
Norepinephrine (20)
Proton pump (19)
ATPase (19)
iGluR (19)
Androgen Receptor (19)
FLT (18)
FGFR (17)
HSV (17)
HDAC (17)
JAK (17)
DNA Alkylator/Crosslinker (17)
RAAS (17)
Bcr-Abl (16)
Src (15)
Adenosine Receptor (15)
Virus Protease (15)
c-Met/HGFR (15)
Opioid Receptor (15)
TRP/TRPV Channel (14)
HBV (14)
Tyrosine Kinases (14)
Progesterone Receptor (13)
PKC (12)
CDK (12)
Raf (12)
TNF (12)
GNRH Receptor (12)
NMDAR (11)
DHFR (11)
Retinoid Receptor (11)
SGLT (11)
ROS (11)
MAO (11)
ALK (11)
HMG-CoA Reductase (10)
Drug Metabolite (10)
Antifolate (10)
P-gp (10)
Reverse Transcriptase (10)
Carbonic Anhydrase (10)
MRP (10)
PARP (10)
AChE (10)
Phosphatase (9)
c-RET (9)
AMPK (9)
Proteasome (9)
Antifection (9)
HCV Protease (9)
mTOR (8)
BTK (8)
HIF/HIF Prolyl-Hydroxylase (8)
CaMK (8)
Lipoxygenase (8)
GluR (8)
DNA Alkylation (8)
MMP (8)
Monoamine Oxidase (8)
P2Y Receptor (8)
PI3K (8)
Phospholipase (7)
Monoamine Transporter (7)
Chloride channel (7)
TAM Receptor (7)
STAT (7)
NADPH (7)
Thrombin (7)
Guanylate cyclase (7)
CFTR (7)
GPR (7)
Trk receptor (7)
ABC (7)
MEK (7)
HER (7)
BCL (6)
Interleukin (6)
DNA Methyltransferase (6)
Neurokinin receptor (6)
IL Receptor (6)
Transferase (6)
Hedgehog/Smoothened (6)
Aromatase (6)
P2X Receptor (6)
ERK (6)
S1P Receptor (6)
Mitochondrial Metabolism (6)
TLR (5)
Endothelin Receptor (5)
Nrf2 (5)
Glutathione Peroxidase (5)
HIF (5)
Akt (5)
DNA (5)
PKA (5)
ribosome (5)
Histone Methyltransferase (5)
LPL Receptor (5)
Vasopressin Receptor (5)
Ras (5)
FXR (5)
Caspase (5)
ROCK (5)
ROS Kinase (5)
PGE Synthase (4)
DPP-4 (4)
GPCR19 (4)
Oxytocin Receptor (4)
HSP (4)
NOD (4)
Amino Acids and Derivatives (4)
Antiviral (4)
Smo (4)
Tyrosinase (4)
Melatonin Receptor (4)
p38 MAPK (4)
GSK-3 (4)
Sigma receptor (4)
NO Synthase (4)
Fatty Acid Synthase (4)
CaSR (4)
IκB/IKK (4)
Wnt/beta-catenin (4)
Beta Amyloid (4)
Antioxidant (4)
Annexin A (4)
FAK (3)
Gamma-secretase (3)
AhR (3)
CXCR (3)
Integrin (3)
cholecystokinin (3)
Aminopeptidase (3)
Leukotriene Receptor (3)
GST (3)
c-Fms (3)
Cysteine Protease (3)
IGF-1R (3)
Ligand for E3 Ligase (3)
Melanocortin Receptor (3)
Adenosine deaminase (3)
Free radical scavengers (3)
Molecular Glues (3)
Isocitrate Dehydrogenase (IDH) (3)
TGF-beta/Smad (3)
Serine/threonin kinase (3)
Na-K-Cl cotransporter (3)
Serine Protease (3)
PAK (3)
MT Receptor (3)
Xanthine Oxidase (3)
UGT (3)
Syk (3)
Hydroxylase (3)
Arginase (2)
Cannabinoid Receptor (2)
Monocarboxylate transporter (2)
CRM1 (2)
Gap Junction Protein (2)
CGRP Receptor (2)
GHSR (2)
CAT (2)
PLK (2)
NOD-like Receptor (NLR) (2)
Cell wall (2)
Protease-activated Receptor (2)
NOS (2)
Reductase (2)
RSV (2)
ROR (2)
Ligands for Target Protein for PROTAC (2)
Beta-Secretase (2)
LTR (2)
Hexokinase (2)
CCR (2)
Decarboxylase (2)
IRE1 (2)
LDL (2)
YAP (2)
Rho (2)
Lipid (2)
IFNAR (2)
MAPK (2)
OAT (2)
Somatostatin (2)
Aryl Hydrocarbon Receptor (2)
Ephrin Receptor (2)
Aurora Kinase (2)
DNA gyrase (2)
NADPH-oxidase (1)
IAP (1)
Chk (1)
Platelet aggregation (1)
cAMP (1)
Bradykinin Receptor (1)
GRK (1)
S6 Kinase (1)
Adiponectin receptor (1)
Glucagon Receptor (1)
Epigenetic Reader Domain (1)
MTH1 (1)
PAFR (1)
CSF-1R (1)
Immunology/Inflammation related (1)
p53 (1)
Imidazoline Receptor (1)
PD-1/PD-L1 (1)
Liver X Receptor (1)
Thrombopoietin Receptor (1)
PDK (1)
Complement System (1)
OX Receptor (1)
Thyroid hormone receptor(THR) (1)
Neprilysin (1)
NPC1L1 (1)
Pyroptosis (1)
GluCls (1)
TOPK (1)
Hydrogenase (1)
JNK (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
ACK (1)
PAD (1)
RAR/RXR  (1)
DUB (1)
FAAH (1)
BACE (1)
PROTAC Linker (1)
Sirtuin (1)
Na+/Ca2+ Exchanger (1)
Histone Demethylase (1)
Lipase (1)
Glutathione reductase (1)
Mdm2 (1)
Factor Xa (1)
ATP Citrate Lyase (1)
VDA (1)
Hck (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
CORPORATE
About Us Careers Privacy Notice Events & News Terms & Conditions
SUPPORT
Contact Us Worldwide Distributors Quality Control Technical Support
RESOURCE
Product Catalog Product Citations Signaling Pathways Solution Calculators
FOLLOW OUR
Social Network
Newsletter Subscription
Subscribe to receive our lastest product updates and special offers!
Corporate
Support
Resource
Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
TargetMol
Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved.