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Search Result

Search Results for " herg "

Targets

HER Melanin-concentrating Hormone Receptor (MCHR)

103

Compounds

9

Natural Products

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T11966 MCHR1 antagonist 2 HER , Melanin-concentrating Hormone Receptor (MCHR)
MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.
T9687 MAGL-IN-4 His121 ARG57 Lipase
MAGL-IN-4 (His121 ARG57) is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.
T1434 Clarithromycin A-56268 P450 , ribosome , MRP , Antibacterial , Antibiotic , Autophagy
Clarithromycin (A-56268) is a Macrolide Antimicrobial. The mechanism of action of clarithromycin is as a Cytochrome P450 3A4 Inhibitor, and Cytochrome P450 3A Inhibitor, and P-Glycoprotein Inhibitor. The chemical classif...
T1496 Amiodarone hydrochloride Amiodar,Amiodarone HCl,Nexterone Potassium Channel , Adrenergic Receptor , Autophagy
Amiodarone hydrochloride (Amiodarone HCl) is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting POTASSIUM CHANNELS and VOLTAGE-GATED SODIUM C...
T1278 Astemizole Laridal,Histaminos,Paralergin Potassium Channel , Histamine Receptor
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re...
T9009 ICA-105574 ICA,3-nitro-N-[4-phenoxyphenyl]-benzamide HER
ICA-105574 (ICA) is an activator of hERG that binds to the channel to remove inactivation, thus increasing peak current amplitude and shortening the action potential. It also modulates activation kinetics of the channel.
T4641 Branaplam LMI 070,NVS-SM1 Others , Potassium Channel , DNA/RNA Synthesis
Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.
T4478 CID 16020046 C390-0219 Cannabinoid Receptor
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
T7198 E-4031 EGFR , Potassium Channel
E-4031 is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by blocking ERG K+ channels (IC50 = 29 nM)
T1676 Rosuvastatin ZD 4522 Potassium Channel , HMG-CoA Reductase , Autophagy
Rosuvastatin (ZD 4522) is an antilipemic agent that competitively inhibits hydroxymethyl-glutaryl-coenzyme A (HMG-CoA) reductase. HMG-CoA reductase catalyzes the conversion of HMG-CoA to mevalonic acid, the rate-limiting...
T1291 Cisapride Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase Potassium Channel , 5-HT Receptor , HER
Cisapride (R 51619) is a serotonin type 4 (5-HT4) receptor agonists are potent prokinetic agents that act on serotonin receptors in the intestine and promote intestinal peristalsis, increase gastric emptying and decrease...
T1510 Rosuvastatin calcium ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium Potassium Channel , HMG-CoA Reductase , Autophagy
Rosuvastatin calcium (ZD4522) , a selective and competitive inhibitor of hepatic hydroxymethyl-glutaryl coenzyme A (HMG-CoA) reductase, has antilipidemic activity.
T16444 PD-118057 Potassium Channel , HER
PD-118057 is a potent ether associated (hERG) potassium channel activator that shows no activity against hERG. PD-118057 inhibits the excitability of the membrane by activating the hERG channel. PD-118057 is a potential ...
T13619 Cloperastine fendizoate Hustazol EGFR
Cloperastine fendizoate (Hustazol) inhibits the hERG K+ currents in a concentration-dependent manner (IC50: 27 nM).
T7195 GSK369796 Dihydrochloride N-tert-butylisoquine Potassium Channel , Parasite
GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate. is an affordable and effective antimalarial and inhibits hERG potassium ion channel repolarization(IC50 of 7.5 μM)
T14077 A-935142 EGFR
A-935142 is a human ether-a-go-go-related gene (hERG, Kv 11.1) channel activator. a-935142 enhances hERG currents by slowing inactivation, promoting activation, reducing inactivation, shortening atrial and ventricular re...
T27117 DA-6886 DA6886,DA 6886 5-HT Receptor
DA-6886 is an agonist 5-Hydroxytryptamine receptor 4 (5-HT4). DA-6886 induced relaxation of the rat oesophagus preparation in a 5-HT4 receptor antagonist-sensitive manner. The evaluation of DA-6886 in CHO cells expressin...
T2641 KRCA-0008 KRCA 0008,KRCA0008 ACK , ALK
KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.
T3192 NS1643 Potassium Channel , HER , Autophagy
NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator with EC50 of 10.5 μM.
TQ0139 VU 0240551 N-(4-Methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide,VU0240551-2-D4 Potassium Channel , Calcium Channel , HER
VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.
T27795L (Iso)-Landipirdine (Iso)-SYN120,(Iso)-RO5025181,(Iso)-Landipirdine(Iso-1000308-25-7) 5-HT Receptor
(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist. (Iso)-Landipirdine has a significant effect on the hERG pharmacophore and can be used to study neurological disorders in the Alzheimer's di...
T10335 Antihistamine-1 P450
Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).
T9146 Ms48107 Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro- Others
MS48107 is a potent, selective positive allosteric modulator of G protein-coupled receptor 68 (GPR68), demonstrating specificity for GPR68 over closely related proton GPCRs, neurotransmitter transporters, and hERG ion ch...
T6175 ADL-5859 ADL5859 Hydrochloride,ADL5859 HCl Opioid Receptor
ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the hERG channel.
T30260 AZD-5672 AZD 5672,AZD5672,UNII-61XQN688TW HER , P-gp , CCR
AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM. AZD-5672 inhibits hERG cardiac ion channel binding and P-gp-mediated digoxin transport with IC50s of 7.3 μM and 32 μM. AZD-5672 can be used in studies about rheu...
T6245 BAPTA-AM BAPTA/AM Potassium Channel
BAPTA-AM is a calcium chelator that is cell-permeable and selective, blocking hERG, hKv1.3, and hKv1.5 channels (IC50=1.3/1.45/1.23 μM). BAPTA-AM has a 105-fold higher affinity for Ca2+ than for Mg2+, and can be used for...
T16265 Naluzotan PRX 00023 EGFR , 5-HT Receptor
Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+ channel blocker with an IC50 value of 3800 nM.Naluzotan exhi...
T12912 Sigma-1 receptor antagonist 3 Sigma receptor , HER
Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain.
T6365 A 922500 A922500,DGAT-1 Inhibitor 4a Acyltransferase , Transferase
A 922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.
T0723 Cloperastine hydrochloride HT-11 hydrochloride Potassium Channel , 5-HT Receptor
Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.
T32191 Irdabisant CEP-26401,CEP 26401,CEP26401 Histamine Receptor
Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R Ki= 7.2 nM, human H3R Ki= 2.0 nM). Irdabisant ex...
T73447 NP10679
NP10679 is a selective, pH dependent GluN2B subunit -specific N-methyl-D-aspartate ( NMDA ) receptor inhibitor with high oral bioavailability and good brain penetration. NP10679 inhibits GluN2B with IC 50 s of 23 and 142...
T4341 Betrixaban PRT054021 Factor Xa
Betrixaban (PRT054021) is a non-vitamin K oral anticoagulant whose action is driven by the competitive and reversible inhibition of the factor Xa [1]. It was selected among all lead compounds due to its low hERG channel ...
T2170 SKF-96365 hydrochloride SKF96365 Apoptosis , Potassium Channel , Calcium Channel , TRP/TRPV Channel , Autophagy
SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y cells. SKF-96365 hydrochloride can induce cytoprotective autopha...
T68113 Naluzotan hydrochloride PRX 00023 hydrochloride EGFR , 5-HT Receptor
Naluzotan hydrochloride (PRX 00023 hydrochloride) is a hERG K+ channel blocker with an IC50 value of 3800 nM and is commonly used in the study of anxiety and depression.Naluzotan hydrochloride is also a novel, potent, an...
T68599 Orphenadrine Orphenadrine (free base) Sodium Channel , NMDAR , AChR
Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner, producing an IC of 0.85 μM in HEK cells.Orphenadrine is an antagoni...
T6618 Orphenadrine Citrate Flexon,Flexoject,Banflex AChR , iGluR
Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.
T11394 GFB-8438 TRP/TRPV Channel
GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).
T7502 PF 05089771 tosylate Sodium Channel
PF-05089771 is a voltage-gated sodium channel 1.7 (Nav1.7) blocker (IC50: 11, 16, 33, and 20 nM for 5N11S, 5A11L, 5A11S, and 5A11L Nav1.7 splice variants, respectively). It is selective for Nav1.7 over Nav1.1-1.6 and 1.8...
T2280 Endoxifen (Z-isomer) Endoxifen Z-isomer Estrogen Receptor/ERR , EGFR , Potassium Channel , Estrogen/progestogen Receptor , HER
Endoxifen Z-isomer (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.
T3215 JNJ-42165279 JNJ42165279 FAAH , Autophagy
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279 (10 μM) exhibits high selectivity against a panel of 50 re...
T4612 NS309 EGFR , Potassium Channel , HER
NS309 is a nonselective activator of small- and intermediate-conductance Ca2+-activated K+ (SK/KCa2 and IK/KCa3.1) channels (EC50s range from 0.12-1.2 µM for SK channels and 10-90 nM for IK channels). It can also activat...
T1266 Terfenadine (±)-Terfenadine,MDL-991 Apoptosis , Potassium Channel , 5-HT Receptor , Caspase , Na+/Ca2+ Exchanger , HER , AChR , Histamine Receptor
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects.
T1066 Ketanserin R41468,Ketanserin tartrate,Ketanserinum Potassium Channel , 5-HT Receptor , Autophagy
Ketanserin (Ketanserinum) is a quinazoline derivative and serotonin (5-hydroxytryptamine, 5HT) receptor subtype 2 (5-HTR2) antagonist with potential antihypertensive and antiplatelet activities. Following administration,...
T34616 Seridopidine ACR-343,ACR 343,ACR343 Dopamine Receptor
Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.
T1066L Ketanserin tartrate KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist with antihypertensive activity, inhibits serotonin-induced vasoconstriction and platelet activation, and can be used in th...
T1320 Disopyramide Triombrin,Hypaque sodium,amidotrizoate sodium Potassium Channel , Sodium Channel , AChR
Disopyramide (Triombrin) is a class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the h...
T4980 Betrixaban maleate Factor Xa
Betrixaban maleate is a non-vitamin K oral anticoagulant whose action is driven by the competitive and reversible inhibition of the factor Xa.
T28347 PD-307243 PD307243
PD-307243 is an activator of hERG channel.
T63430 Rosuvastatin Sodium
Rosuvastatin Sodium is a competitive HMG-CoA reductase (HMGCR) inhibitor (IC50: 11 nM) that effectively blocks hERG currents (IC50: 195 nM). Rosuvastatin Sodium reduces the expression of mature hERG and inhibits the inte...

Compounds

MCHR1 antagonist 2
T11966
Synonym:
Target: HER, Melanin-concentrating Hormone Receptor (MCHR)
MAGL-IN-4
T9687
Synonym: His121 ARG57
Target: Lipase
Clarithromycin
T1434
Synonym: A-56268
Target: P450, ribosome, MRP, Antibacterial, Antibiotic, Autophagy
Amiodarone hydrochloride
T1496
Synonym: Amiodar,Amiodarone HCl,Nexterone
Target: Potassium Channel, Adrenergic Receptor, Autophagy
Astemizole
T1278
Synonym: Laridal,Histaminos,Paralergin
Target: Potassium Channel, Histamine Receptor
ICA-105574
T9009
Synonym: ICA,3-nitro-N-[4-phenoxyphenyl]-benzamide
Target: HER
Branaplam
T4641
Synonym: LMI 070,NVS-SM1
Target: Others, Potassium Channel, DNA/RNA Synthesis
CID 16020046
T4478
Synonym: C390-0219
Target: Cannabinoid Receptor
E-4031
T7198
Synonym:
Target: EGFR, Potassium Channel
Rosuvastatin
T1676
Synonym: ZD 4522
Target: Potassium Channel, HMG-CoA Reductase, Autophagy
Cisapride
T1291
Synonym: Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase
Target: Potassium Channel, 5-HT Receptor, HER
Rosuvastatin calcium
T1510
Synonym: ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium
Target: Potassium Channel, HMG-CoA Reductase, Autophagy
PD-118057
T16444
Synonym:
Target: Potassium Channel, HER
Cloperastine fendizoate
T13619
Synonym: Hustazol
Target: EGFR
GSK369796 Dihydrochloride
T7195
Synonym: N-tert-butylisoquine
Target: Potassium Channel, Parasite
A-935142
T14077
Synonym:
Target: EGFR
DA-6886
T27117
Synonym: DA6886,DA 6886
Target: 5-HT Receptor
KRCA-0008
T2641
Synonym: KRCA 0008,KRCA0008
Target: ACK, ALK
NS1643
T3192
Synonym:
Target: Potassium Channel, HER, Autophagy
VU 0240551
TQ0139
Synonym: N-(4-Methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide,VU0240551-2-D4
Target: Potassium Channel, Calcium Channel, HER
(Iso)-Landipirdine
T27795L
Synonym: (Iso)-SYN120,(Iso)-RO5025181,(Iso)-Landipirdine(Iso-1000308-25-7)
Target: 5-HT Receptor
Antihistamine-1
T10335
Synonym:
Target: P450
ms48107
T9146
Synonym: Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro-
Target: Others
ADL-5859
T6175
Synonym: ADL5859 Hydrochloride,ADL5859 HCl
Target: Opioid Receptor
AZD-5672
T30260
Synonym: AZD 5672,AZD5672,UNII-61XQN688TW
Target: HER, P-gp, CCR
BAPTA-AM
T6245
Synonym: BAPTA/AM
Target: Potassium Channel
Naluzotan
T16265
Synonym: PRX 00023
Target: EGFR, 5-HT Receptor
Sigma-1 receptor antagonist 3
T12912
Synonym:
Target: Sigma receptor, HER
A 922500
T6365
Synonym: A922500,DGAT-1 Inhibitor 4a
Target: Acyltransferase, Transferase
Cloperastine hydrochloride
T0723
Synonym: HT-11 hydrochloride
Target: Potassium Channel, 5-HT Receptor
Irdabisant
T32191
Synonym: CEP-26401,CEP 26401,CEP26401
Target: Histamine Receptor
NP10679
T73447
Synonym:
Target:
Betrixaban
T4341
Synonym: PRT054021
Target: Factor Xa
SKF-96365 hydrochloride
T2170
Synonym: SKF96365
Target: Apoptosis, Potassium Channel, Calcium Channel, TRP/TRPV Channel, Autophagy
Naluzotan hydrochloride
T68113
Synonym: PRX 00023 hydrochloride
Target: EGFR, 5-HT Receptor
Orphenadrine
T68599
Synonym: Orphenadrine (free base)
Target: Sodium Channel, NMDAR, AChR
Orphenadrine Citrate
T6618
Synonym: Flexon,Flexoject,Banflex
Target: AChR, iGluR
GFB-8438
T11394
Synonym:
Target: TRP/TRPV Channel
PF 05089771 tosylate
T7502
Synonym:
Target: Sodium Channel
Endoxifen (Z-isomer)
T2280
Synonym: Endoxifen Z-isomer
Target: Estrogen Receptor/ERR, EGFR, Potassium Channel, Estrogen/progestogen Receptor, HER
JNJ-42165279
T3215
Synonym: JNJ42165279
Target: FAAH, Autophagy
NS309
T4612
Synonym:
Target: EGFR, Potassium Channel, HER
Terfenadine
T1266
Synonym: (±)-Terfenadine,MDL-991
Target: Apoptosis, Potassium Channel, 5-HT Receptor, Caspase, Na+/Ca2+ Exchanger, HER, AChR, Histamine Receptor
Ketanserin
T1066
Synonym: R41468,Ketanserin tartrate,Ketanserinum
Target: Potassium Channel, 5-HT Receptor, Autophagy
Seridopidine
T34616
Synonym: ACR-343,ACR 343,ACR343
Target: Dopamine Receptor
Ketanserin tartrate
T1066L
Synonym: KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate
Target: 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
Disopyramide
T1320
Synonym: Triombrin,Hypaque sodium,amidotrizoate sodium
Target: Potassium Channel, Sodium Channel, AChR
Betrixaban maleate
T4980
Synonym:
Target: Factor Xa
PD-307243
T28347
Synonym: PD307243
Target:
Rosuvastatin Sodium
T63430
Synonym:
Target:
1 2 3
Cat No. Product Name Synonyms Targets
T0801 Tannic acid Gallotannic acid Potassium Channel , HER , CXCR
Tannic acid (Gallotannic acid) is a novel hERG channel blocker.
T3054 Daurisoline (R,R)-Daurisoline Others , Potassium Channel , Autophagy
Daurisoline ((R,R)-Daurisoline) is a hERG inhibitor. Daurisoline is also an autophagy blocker.
TN1092 O-Nornuciferine Potassium Channel , HER
O-Nornuciferine reveals distinct in vitro hERG blockages measured in HEK293 cells with the IC50 value of 2.89 uM.
T8189 Dihydroberberine Potassium Channel , HSP , HER
Dihydroberberine has anti-atherosclerotic, anti-inflammatory, hypolipidemic and antitumor activities. It inhibits human ether-a-go-go-related gene (hERG) channels and remarkably reduces Hsp90 expression and its interacti...
T8182 Guanfu base A Guan-fu base A P450 , Potassium Channel , HER
Guanfu base A is a potent noncompetitive CYP2D6 inhibitor (Ki: 1.20 μM in HLMs; Ki: 0.37 μM for rCYP2D6). It also inhibits HERG channel current.
T3A2467 Allocryptopine Thalictrimine,Fagarine I Potassium Channel
Allocryptopine (Thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively.
T4550 Ajmaline Cardiorythmine,Raugalline,Tachmalin,(+)-Ajmaline Sodium Channel
Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and...
TN6051 Songoramine
Songoramine(10 uM) demonstrates significant hERG K+ channel inhibition.
TN4638 Neolinine EGFR , Potassium Channel
Neolinine(at 10uM) shows significant hERG K+ channel inhibition activity.

Natural Products

Tannic acid
T0801
Synonym: Gallotannic acid
Target: Potassium Channel, HER, CXCR
Daurisoline
T3054
Synonym: (R,R)-Daurisoline
Target: Others, Potassium Channel, Autophagy
O-Nornuciferine
TN1092
Synonym:
Target: Potassium Channel, HER
Dihydroberberine
T8189
Synonym:
Target: Potassium Channel, HSP, HER
Guanfu base A
T8182
Synonym: Guan-fu base A
Target: P450, Potassium Channel, HER
Allocryptopine
T3A2467
Synonym: Thalictrimine,Fagarine I
Target: Potassium Channel
Ajmaline
T4550
Synonym: Cardiorythmine,Raugalline,Tachmalin,(+)-Ajmaline
Target: Sodium Channel
Songoramine
TN6051
Synonym:
Target:
Neolinine
TN4638
Synonym:
Target: EGFR, Potassium Channel

Recombinant Proteins

Species：
Human (2)
Expression System：
Baculovirus-Insect Cells (1)
in vitro E. coli expression system (1)
Tag：
His,GST (1)
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPY-04561 SGK3 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
Serine / threonine-protein kinase Sgk3, also known as Serum / glucocorticoid-regulated kinase 3, Serum / glucocorticoid-regulated kinase-like and SGK3, is a cytoplasmic vesicle protein that belongs to the protein kinase ...
TMPH-01891 KCNE2 Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Ancillary protein that assembles as a beta subunit with a voltage-gated potassium channel complex of pore-forming alpha subunits. Modulates the gating kinetics and enhances stability of the channel complex. Assembled wit...
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