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Results for "

gpr88

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    10
    TargetMol | Inhibitors_Agonists
GPR88-IN-1
T79901714265-50-6
GPR88-IN-1 is a GPR88 antagonist that can be used for researching central nervous system disorders [1].
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8-10 weeks
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GPR88 agonist 2
T79902
GPR88 agonist 2 (compound 53) is a potent, brain-penetrant agonist of GPR88, with an EC50 of 14 µM in the GPR88 cAMP functional assay [1].
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GPR88 agonist 3
T865222963597-44-4
GPR88 agonist 3 (compound 20), exhibiting an EC50 of 204 nM, functions as an agonist for GPR88. It is applicable in the research of psychiatric and neurodegenerative disorders [1].
  • Inquiry Price
6-8 weeks
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(1R,2R)-2-PCCA hydrochloride
(1R,2R)-2-PCCA(hydrochloride)
T134231609563-71-4In house
(1R,2R)-2-PCCA hydrochloride is a potent, selective, and blood-brain-barrier-crossing GPR88 receptor agonist with an EC50 value of 1140 n in striatal membranes of WT mice; it can be used to study the central nervous system.
  • Inquiry Price
6-8 weeks
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(1S,2R)-2-PCCA
(1S,2R)-2-PCCA(Iso-1609563-71-4)
T13423L In house
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value of 3 nM in the non-cellular system and 603 nM in the cellular system.
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TargetMol | Inhibitor Sale
2-PCCA hydrochloride
2-PCCA hydrochloride(1609624-97-6 Free base)
T806661609563-70-3In house
2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of GPR88-mediated cAMP production in HEK293 cells with an EC50 value of 116 nM.
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RTI-13951-33 hydrochloride
RTI-13951-33 hydrochloride (2244884-08-8 free base)
T12778
RTI-13951-33 hydrochloride is a potent, selective, and brain-penetrant GPR88 agonist, exhibiting an EC50 of 25 nM in vitro cAMP functional assay. It significantly reduces alcohol reinforcement and intake behaviors in rats [1].
  • Inquiry Price
3-6 months
Size
QTY
RTI-13951-33
T12778L2244884-08-8
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).
  • Inquiry Price
8-10 weeks
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RTI-122
T2008643034664-39-3
RTI-122 is an effective GPR88 agonist with good metabolic stability (half-life of 5.8 hours in mice) and a cAMP EC50 of 11 nM. It can penetrate the blood-brain barrier and is utilized in research related to excessive drinking.
  • Inquiry Price
3-6 months
Size
QTY
2-PCCA
T710541287205-42-8
2-PCCA is a GPR88 agonist.
  • Inquiry Price
1-2 weeks
Size
QTY