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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9744 | MP07-66 | Phosphatase | |
MP07-66 is a novel FTY720-analog devoid of immunosuppressive effects leads to the reactivation of PP2A, which in turn triggers apoptosis of CLL cells. | |||
T4007 | Eticlopride hydrochloride | Dopamine Receptor | |
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM). | |||
T9933 | Methyl 2,4-dihydroxyphenylacetate | Others | |
Methyl 2,4-dihydroxyphenylacetate is a natural product isolated from Nigella damascena seeds with selective phytotoxic effects. | |||
TN5634 | Aureusidin | Auresudidin,Auresidin | Antioxidant , Reactive Oxygen Species , Lipoxygenase |
Aureusidin (Auresidin) shows antioxidant and lipoxygenase inhibitory activity with anti-inflammatory effects. | |||
T5648 | Purpurin | 1,2,4-Trihydroxyanthraquinone,Hydroxylizaric acid,Verantin | MAO , Antibacterial , Antibiotic , Antifungal |
Purpurin (Verantin) was a reversible and competitive inhibitor of MAO-A with a Ki value of 0.422μM. it exhibits anti-angiogenic, antifungal, antibiotic, and antioxidative activities. | |||
T15286 | Flindokalner | BMS-204352 | Potassium Channel |
Flindokalner (BMS-204352) is a potassium channel modulator and a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is a large conductance calcium-activated K channel (BKca) p... | |||
T2009 | SB-3CT | MMP | |
SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM). | |||
T13741 | Isoviolanthin | Others | |
Isoviolanthin reduces the migratory and invasive capacities of TGF-β1-treated HCC cells without cytotoxic effects on normal live cells and has potential as a therapeutic agent for the treatment of advanced-stage metastat... | |||
T3858 | Macranthoidin A | Others | |
Macranthoidin A has anti-inflammation activity. | |||
T9461 | AZ194 | Sodium Channel | |
CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor. | |||
T8014 | Epoxylinalool | 2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran | Others |
Epoxylinalool (2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran) is a naturally occurring monoterpene alcohol widely used in the production of perfumes and flavors. | |||
T8516 | Levomenol | (-)-α-BISABOLOL | Others |
Levomenol ((-)-α-BISABOLOL) is a sesquiterpene alcohol that has been found in the essential oils of several aromatic plants, with exerts antioxidant, anti-inflammatory, and anti-apoptotic activities. | |||
T19916 | TRIM | 1-(2-Trifluoromethylphenyl)imidazole | NOS |
TRIM (1-(2-Trifluoromethylphenyl)imidazole) is an inhibitor of nNOS. | |||
T0389 | Dabigatran etexilate | BIBR 1048 | Thrombin |
Dabigatran etexilate (BIBR 1048) is a thrombin inhibitor, which acts by binding and blocking thrombogenic activity and the prevention of thrombus formation. | |||
T5133 | Dabigatran Etexilate Mesylate | BIBR 1048MS,Dabigatran etexilate methanesulfonate | Thrombin |
Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor (DTI, Ki: 4.5 nM). | |||
TP2036 | DPDPE | Opioid Receptor | |
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinociceptive in vivo. | |||
T3026 | (-)-Huperzine A | HupA,Huperzine A | Apoptosis , AChR , AChE , iGluR |
(-)-Huperzine A (HupA) , an active Lycopodium alkaloid extracted from the traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the tr... | |||
T4S0554 | Theaflavine-3,3'-digallate | TFBG,theaflavin digallate | Others |
1. Theaflavine-3,3'-digallate (theaflavin digallate) and lactic acid together could reduce herpes simplex virus transmission. | |||
T3739 | 2,6-Dimethoxyquinone | 2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone | Others |
2,6-Dimethoxyquinone (2,6-Dimethoxy-p-benzoquinone) is a member of the class of compounds known as P-benzoquinones. 2,6-Dimethoxyquinone is slightly soluble (in water) and an extremely weak basic (essentially neutral) co... | |||
T60022 | Aromatase-IN-2 | Others | |
Aromatase-IN-2 has anti-inflammatory, antitumor and antiasthmatic effects. |