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Cat No. | Product Name | Synonyms | Targets |
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T67898 | α-Glucosidase-IN-22 | Glucosidase | |
α-Glucosidase-IN-22 is a selective inhibitor of α-glucosidase (IC50=0.64 μM). α-Glucosidase-IN-22 has antidiabetic activity and has potential in type 2 diabetes (T2DM) studies. | |||
T67728 | α-Glucosidase-IN-23 | Glucosidase | |
α-Glucosidase-IN-23 is an orally active α-Glucosidase inhibitor. α-Glucosidase-IN-23 can decrease blood glucose by α-glucosidase inhibition (IC50= 4.48 μM). | |||
T41028 | α-Glucosidase | α-D-Glucosidase | |
α-Glucosidase (α-D-Glucosidase) is a carbohydrate hydrolyzing enzyme that catalyzes the release of α-glucose from the non-reducing end of the substrate. It plays a vital role in facilitating glucose absorption by the sma... | |||
T60715 | α-Glucosidase-IN-4 | Glucosidase | |
α-Glucosidase-IN-4 is a potent α-glucosidase inhibitor with antihypertensive and hypoglycemic activity. | |||
T76110 | β-Glucosidase | ||
β-Glucosidase, a pivotal enzyme in cellulose degradation, belongs to the extensive family of glycoside hydrolases. It plays a crucial role in breaking down cellulose in soils and holds promise for assessing biological so... | |||
T63562 | α-Glucosidase-IN-14 | ||
α-Glucosidase-IN-14 is a potent inhibitor of α-glucosidase (IC50: 5.22 μM). | |||
T62222 | α-Glucosidase-IN-11 | ||
α-Glucosidase-IN-11 is a highly permeable competitive inhibitor of α-glucosidase (IC50: 0.56 μM). α-Glucosidase-IN-11 binds to the Trp residue in α-glucosidase and has a regulatory effect on protein folding and can be us... | |||
T61519 | α-Glucosidase-IN-18 | ||
α-Glucosidase-IN-18 (7B) is an orally active inhibitor of α-glucosidase, displaying an IC 50 value of 3.96 μM. This compound exhibits antidiabetic properties [1]. | |||
T61166 | α-Glucosidase-IN-16 | ||
α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM. This compound demonstrates the ability to significantly decrease blood glucose ... | |||
T61124 | α-Glucosidase-IN-9 | ||
α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1]. | |||
T60389 | α-Glucosidase-IN-5 | ||
α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM. α-Glucosidase-IN-5 has the potential for the research of diabete... | |||
T79237 | α-Glucosidase-IN-27 | Glucosidase | |
α-Glucosidase-IN-27 (compound 8l), an α-glucosidase inhibitor with an IC50 value of 25.78 μM, demonstrates potential for research into type 2 diabetes (D2M) [1]. | |||
T78794 | α-Glucosidase-IN-31 | Glucosidase | |
α-Glucosidase-IN-31 (compound R1) is a potent oral α-Glucosidase inhibitor with an IC50 of 10.1 μM, demonstrating significant blood glucose reduction and antidiabetic activity [1]. | |||
T79700 | α-Glucosidase-IN-32 | Glucosidase | |
α-Glucosidase-IN-32 (compound f26) is a reversible, noncompetitive inhibitor of α-glucosidase that is orally active and exhibits an IC50 of 3.07 μM. It forms a complex with α-glucosidase via hydrogen bonding and hydropho... | |||
T80709 | α-Glucosidase-IN-41 | Glucosidase | |
α-Glucosidase-IN-41 (compound 5o), a potent inhibitor of α-glucosidase, induces alterations in the secondary structure of the enzyme, thereby impeding its catalytic function. This compound is utilized in the study of dia... | |||
T78740 | α-Glucosidase-IN-28 | Glucosidase | |
α-Glucosidase-IN-28 (Compound 18) is an α-glucosidase inhibitor with an IC50 of 0.62 μM and Ki value of 3.93 μM. It interacts with the enzyme's original binding site (OBS) and establishes multiple hydrophobic interaction... | |||
T63310 | α-Glucosidase-IN-6 | ||
α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies. | |||
T61503 | α-Glucosidase-IN-15 | ||
α-Glucosidase-IN-15 (Compound 14B) exhibits potent inhibitory activity against α-glucosidase, with an IC50 value of 3.34 μM. It possesses antidiabetic properties [1]. | |||
T62972 | α-Glucosidase-IN-17 | ||
α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitory concentration (IC50) of 3.79 μM [1]. | |||
T80711 | α-Glucosidase-IN-39 | Glucosidase | |
α-Glucosidase-IN-39 is a potent α-glucosidase enzyme inhibitor, exhibiting an IC50 value of 869.06 ppm. It is applicable for use in antidiabetic studies [1]. | |||
T61761 | α-Glucosidase-IN-21 | ||
α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase. With an impressive IC50 value of 2.62 μM, this compound exhibits remarkable anti-diabetic properties [1]. | |||
T61331 | α-Glucosidase-IN-20 | ||
α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase. It exhibits potent anti-diabetic properties, as evidenced by its IC50 value of 3.01 μM [1]. | |||
T78864 | α-Glucosidase-IN-33 | Glucosidase | |
α-Glucosidase-IN-33 (compound 7c), with an IC50 of 2.39 μM, is a potent inhibitor of α-glucosidase and is relevant in research on type 2 diabetes and hyperglycemia [1]. | |||
T78865 | α-Glucosidase-IN-34 | Glucosidase | |
α-Glucosidase-IN-34 (compound 7f) is a potent inhibitor of α-glucosidase, exhibiting an IC50 of 2.90 μM, and is applicable in research related to type 2 diabetes and hyperglycemia [1]. | |||
T80708 | α-Glucosidase-IN-42 | Glucosidase | |
α-Glucosidase-IN-42 (Compound 26), a 9-O-berberrubine carboxylate derivative, exhibits potent α-glucosidase inhibitory activity with an IC50 value of 1.61 μM and has potential for use in antidiabetic research [1]. | |||
T78741 | α-Glucosidase-IN-29 | Glucosidase | |
α-Glucosidase-IN-29 (compound 19) is an inhibitor of α-glucosidases, exhibiting an IC50 value of 1.21 μM and a Ki of 1.80 μM. This compound is utilized in the research of diabetes and related diseases [1]. | |||
T63361 | α-Glucosidase-IN-13 | ||
α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM). | |||
T62994 | α-Glucosidase-IN-10 | ||
α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes. | |||
T63574 | α-Glucosidase-IN-12 | ||
α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM). | |||
T61249 | α-Glucosidase-IN-2 | ||
α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an antidiabetic agent [1]. | |||
T62891 | α-Glucosidase-IN-19 | ||
Alpha-Glucosidase-IN-19 (Compound 6B) is an orally active alpha-glucosidase inhibitor (IC50: 3.63 μM) with antidiabetic effects. | |||
T61094 | α-Glucosidase-IN-8 | ||
α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1]. | |||
T64230 | α-Glucosidase-IN-3 | ||
α-Glucosidase-IN-3 is an oleanolic acid oxime ester derivative targeting α-glucosidase and α-amylase with an IC50 value of 0.35 μM for α-glucosidase. | |||
T80710 | α-Glucosidase-IN-40 | Glucosidase | |
α-Glucosidase-IN-40 (compound 5) serves as a noncompetitive inhibitor of the α-glucosidase enzyme, exhibiting an inhibitory concentration (IC50) of 24.62 μM [1]. | |||
T80712 | α-Glucosidase-IN-38 | Glucosidase | |
α-Glucosidase-IN-38 (Compound 11j) is a potent α-glucosidase inhibitor, demonstrating an IC50 of 12.44±0.38 μM, and is significant in the context of Diabetes mellitus (DM) management [1]. | |||
T78731 | α-Glucosidase-IN-26 | Glucosidase | |
α-Glucosidase-IN-26 (Compound 7i), with an IC50 value of 4.63 µM, functions as an α-glucosidase inhibitor and is utilized in research related to type 2 diabetes mellitus (T2DM) [1]. | |||
T79259 | α-Glucosidase-IN-25 | Glucosidase | |
α-Glucosidase-IN-25 (Compound (R)-8k) serves as a competitive inhibitor for α-glucosidase, demonstrating an inhibitory concentration 50 (IC50) of 1.19μM, making it applicable in anti-diabetic research [1]. | |||
T78881 | α-Glucosidase-IN-36 | Glucosidase | |
α-Glucosidase-IN-36 (compound 5g) is a potent inhibitor of α-glucosidase, exhibiting an IC50 value of 6.69 ± 0.18 μM and inhibition constants Ki and Kis of 1.65 μM and 4.54 μM, respectively. It is hypothesized to suppres... | |||
T79318 | α-Glucosidase-IN-30 | Glucosidase | |
α-Glucosidase-IN-30 (compound 8c) is a potent, orally active competitive inhibitor of α-glucosidase, exhibiting a K i of 40.0 µM and an IC50 of 49.0 µM. It is non-cytotoxic to both cancerous MCF-7 and normal HDF cell lin... | |||
T61706 | α-Amylase/α-Glucosidase-IN-2 | ||
α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM and 13.09 μM, respectively. This compound shows promise for in... | |||
T79225 | α-Amylase/α-Glucosidase-IN-3 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-3 (Compound 17) serves as a dual inhibitor targeting both α-Amylase and α-Glucosidase, exhibiting IC50 values of 0.70 μM and 1.10 μM, respectively. It is applicable for type-II diabetes mellitu... | |||
T60255 | α-Amylase/α-Glucosidase-IN-1 | ||
α-Amylase/α-Glucosidase-IN-1 (compound 33) is an effective inhibitor of α-amylase/α-glucosidase with IC 50 s of 2.01, 2.09 μM for α-amylase and α-glucosidase, respectively. Kinetic studies predict that α-Amylase/α-Glucos... | |||
T79402 | α-Amylase/α-Glucosidase-IN-4 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-4 (compound 5), a dual inhibitor targeting α-amylase (Amylases) and α-glucosidase (Glucosidase), exhibits potent inhibition with IC50 values of 1.10 μM and 0.15 μM respectively. This compound i... | |||
T80715 | α-Amylase/α-Glucosidase-IN-6 | ||
α-Amylase/α-Glucosidase-IN-6 (compound 5j) serves as a potent dual inhibitor of both α-amylase and α-glucosidase, exhibiting IC50 values of 17.0 µM and 40.1 µM, respectively. It demonstrates anti-hyperglycemic activities... | |||
T78878 | α-Amylase/α-Glucosidase-IN-5 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-5 (compound 4l) functions as a dual inhibitor, effectively inhibiting both α-glucosidase (Glucosidase) and α-amylase (Amylases) with IC50 values of 5.96 μM and 1.62 μM, respectively, exhibiting... | |||
TQ0300 | Conduritol B epoxide | Glucosidase | |
Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase). | |||
T8989 | NCGC 607 | NCGC607 | Others |
NCGC 607 is a a noninhibitory chaperone of glucocerebrosidase (GCase). | |||
T8986 | ML198 | Glucokinase | |
ML198 is a novel activator and non-inhibitory chaperone of glucocerebrosidase. ML198 serves as a starting point to develop a novel approach towards small molecule treatment for patients suffering from Gaucher disease. | |||
T4280 | Gcase activator 1 | LTI-291,LTI 291,LTI291 | Glucosidase |
Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator. | |||
T0920 | Ambroxol | Ambroxolum,NA-872 | P450 , Autophagy |
Ambroxol (NA-872) is a secretolytic agent used in the treatment of respiratory diseases associated with viscid or excessive mucus. It is the active ingredient of Mucosolvan, Lasolvan or Mucoangin. The substance is a muco... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3S0860 | Gitogenin | UGT | |
1. Gitogenin, tigogenin, and solasodine are novel selective inhibitors of UGT1A4, and do not inhibit the activities of major human CYP isoforms. 2. Gitogenin and (25S)-5α-furastan-3β, 22, 26-triol are the inhibitors of e... | |||
T75612 | α-Glucosidase-IN-24 | ||
α-Glucosidase-IN-24 (Compound 13), an α-Glucosidase inhibitor, exhibits an IC50 value of 451 μM and can be derived from Swertia kouitchensis [1]. | |||
T80713 | α-Glucosidase-IN-37 | ||
α-Glucosidase-IN-37 (Compound 11) moderately inhibits lipopolysaccharide (LPS)-induced nitric oxide (NO) production in macrophages, exhibiting an inhibitory concentration 50 (IC50) value of 23.7 μM. Additionally, this co... | |||
T13130 | Terphenyllin | Glucosidase | |
Terphenyllin has α-glucosidase inhibitory activity, and is a natural product isolated from the coral derived fungus Aspergillus candidus. | |||
TN6771 | Malabaricone B | Others | |
Malabaricone B is a Spice-derived phenolic, it induces mitochondrial damage in lung cancer cells via a p53-independent pathway. | |||
T7544 | Fucoidan | Others | |
Fucoidan is found in various species of brown seaweed and algae,with anticancer, antiviral, neuroprotective, immune-modulating. | |||
TN1451 | Brevifolincarboxylic acid | AhR , Aryl Hydrocarbon Receptor , Glucosidase | |
Brevifolincarboxylic acid is a natural product isolated from Polygonum capitatum, it has inhibitory effect on the aryl hydrocarbon receptor (AhR). Brevifolincarboxylic acid is an α-glucosidase inhibitor with an IC50 of 3... | |||
T8319 | Butyl isobutyl phthalate | ButylIsobutylPhthalate | Glucosidase |
Butyl isobutyl phthalate (ButylIsobutylPhthalate) is a non-competitive α-glucosidase inhibitor(IC50 :38 μM),it shows a hypoglycemic effect | |||
TN1990 | Norathyriol | Akt , DNA/RNA Synthesis , AMPK , PPAR | |
Norathyriol is a potent PTP1B inhibitor with good cell permeability and oral availability. | |||
T12142 | N-Caffeoyl O-methyltyramine | Glucosidase | |
N-Caffeoyl O-methyltyramine is isolated from Cuscuta reflexa with strong inhibitory activity against α-glucosidase with IC50 of 103.58 μM. | |||
T41044 | Naringinase | Glucosidase | |
Naringinase is a hydrolytic enzymatic complex that exhibits α-L-rhamnosidase and β-D-glucosidase activities. It is widely found in nature and is primarily utilized for the biotransformation of steroids, antibiotics, and ... | |||
T8260 | 4',5-Dihydroxyflavone | Lipoxygenase , Glucosidase | |
4',5-Dihydroxyflavone is a soybean LOX-1(Ki: 102.6 μM) and yeast α-Glucosidase inhibitor (IC50: 66 μM). | |||
T7028 | Licochalcone C | LICOCHALCONEC | Phosphatase , Antioxidant , Glucosidase |
Licochalcone C (LICOCHALCONEC) has potent antioxidant properties and inhibition of bacterial growth and cellular respiration. It has cardioprotection effect, via antioxidant, anti-inflammatory, and anti-apoptotic activit... | |||
TN2030 | P-Hydroxyphenethyl trans-ferulate | 5-HT Receptor | |
P-Hydroxyphenethyl trans-ferulate exhibits affinity toward 5-HT(7) receptors in a competitive binding assay. P-Hydroxyphenethyl trans-ferulate can double quinone reductase specific activity in Hepa 1c1c7 cells at a level... | |||
T0247 | Acarbose | BAY g 5421 | Glucosidase |
Acarbose (BAY g 5421) is an inhibitor of α-Glucosidases with antihyperglycemic activity. | |||
T2956 | Cedryl acetate | Cedrol acetate,Cedranyl acetate | Antifungal |
Cedryl acetate (Cedranyl acetate) , an acetylated from cedarwood oil, has been applied to chemistry for its properties as a chiral and cell signaling reagent with antifungal and immunotoxicity functions. | |||
T6723 | Voglibose | AO 128,Glustat,Basen | Glucosidase |
Voglibose (Glustat), an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemia and various disorders caused by hyperglycemia. | |||
TN2144 | Resveratroloside | P450 , NO Synthase | |
Resveratroloside has cardioprotective effect, it exhibits α±-glucosidase inhibitory activity, it also can inhibit hydroxylation of testosterone by CYP3A4. | |||
T8202 | Kaempferol 3-O-gentiobioside | Kaempferol 3-gentiobioside | Glucosidase |
Kaempferol 3-O-gentiobioside is a flavonoid isolated from C. alata leaves with antidiabetic activity. It possesses activity against α-glucosidase and displays a carbohydrate enzyme inhibitory effect (IC50: 50 μM). | |||
T2S1158 | 4,5-Dicaffeoylquinic acid | 3,4-Dicaffeoylquinic acid,Isochlorogenic acid C | Others , HBV , Endogenous Metabolite |
1. 4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) has antiviral activity, including anti-HIV-1 integrase activity. 2. 4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) shows anti-hepatotoxic activity. | |||
TN1926 | Methyl caffeate | Methyl caffeate acid | Others , Antibacterial |
Methyl caffeate (Methyl caffeate acid) acid | |||
T5S0788 | Oroxin A | Baicalein 7-O-glucoside | PPAR |
Oroxin A (Baicalein 7-O-glucoside) has antitussive and expectorant effects. | |||
TQ0308 | Castanospermine | 1,6,7,8-Tetrahydroxyoctahydroindolizine,(1S,6S,7R,8R,8aR)-1,6,7,8-Tetrahydroxyindolizidine | Glucosidase |
Castanospermine (1,6,7,8-Tetrahydroxyoctahydroindolizine) is a natural compound that inhibits α- and β-glucosidases, especially glucosidase l. | |||
T3675 | 1-Deoxynojirimycin | Duvoglustat,Moranoline,moranolin | PI3K , Glucosidase |
1-Deoxynojirimycin (Moranoline) is a potent α-glucosidase inhibitor, suppressing postprandial blood glucose, thereby possibly preventing diabetes mellitus. | |||
T6S1525 | 3,4-Dicaffeoylquinic acid | Isochlorogenic acid B | Apoptosis , Antioxidant , Influenza Virus , Endogenous Metabolite |
3,4-Dicaffeoylquinic acid (Isochlorogenic acid B) has antioxidant activity. | |||
T3235 | Rebaudioside A | Reb-A 97,Reb A,Stevioside A3,Glycoside A3 | Endogenous Metabolite , Glucosidase |
Rebaudioside A (Reb A) is a novel agent of glycoside clathration of pharmacons, acts as α-glucosidase inhibitor. | |||
T21344 | 1-Deoxynojirimycin hydrochloride | Moranoline,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin | PI3K , Antibacterial , Antibiotic , Glucosidase |
1-Deoxynojirimycin hydrochloride (Moranoline) is a potent and selective inhibitor of alpha-glucosidase, most commonly found in mulberry leaves. Duvoglustat is used to suppress the elevation of postprandial hyperglycemia. | |||
TN6784 | Ethyl rosmarinate | Methyl rosmarinate | MMP , Tyrosinase , Glucosidase |
Methyl rosmarinate (Methyl rosmarinate) inhibit the activity of tyrosinase, α-glucosidase, and matrix metalloproteinase-1 (MMP-1). | |||
TN2326 | (Z)-Butylidenephthalide | (Z)-3-Butylidenephthalide | Glucosidase |
(Z)-Butylidenephthalide ((Z)-3-Butylidenephthalide) has antitumor and hypoglycemic effects, and can effectively inhibit the tumor growth of glioma and inhibit R-glucosidase activity. | |||
TN1487 | Chrysin 6-C-arabinoside 8-C-glucoside | Others | |
Chrysin 6-C-arabinoside 8-C-glucoside and chrysin-6-C-glucosyl-8-C-arabinoside are α±-glucosidase inhibitors, α±-glucosidase inhibitors are widely used in the treatment of type 2 diabetes. | |||
TN1488 | Chrysin 6-C-glucoside 8-C-arabinoside | Others | |
Chrysin 6-C-glucoside 8-C-arabinoside and Chrysin-6-C-arabinosyl-8-C-glucoside are α±-glucosidase inhibitors, α±-glucosidase inhibitors are widely used in the treatment of type 2 diabetes. | |||
T3S2072 | 3-Butylidenephthalide | Butylidene phthalide,n-Butylidenephthalide | Parasite , Glucosidase |
1. 3-Butylidenephthalide (Butylidene phthalide) has antihyperglycemic effect is due to inhibition of α-glucosidase at the intestinal level, inhibited the activity of yeast-α-glucosidase (IC(5) 2.35 mM) in a noncompetitiv... | |||
TL0009 | Coniferin | Coniferoside,Abietin | Others , Antifungal |
Coniferin (Abietin) has ATP-dependent transport activity and has anti-oxidation effects. Coniferin has preferred substrates for the coniferin beta-glucosidase, the chromogenic coniferin analogue show the exclusive presen... | |||
T1529 | Miglitol | BAY1099,BAY-m1099 | Others |
Miglitol (BAY1099) is an alpha-Glucosidase Inhibitor with antihyperglycemic activity. | |||
TN2302 | Viscidulin III | Ganhuangenin | Glucosidase |
Viscidulin III (Ganhuangenin) is present in Scutellaria baicalensis and acts as an α-glucosidase inhibitor. | |||
T6S2122 | Ginkgolic Acid (C13:0) | 6-Tridecylsalicylic acid,Ginkgolic acid (13:0),Ginkgoneolic Acid,Ginkgolic acid C13:0 | Antibacterial , Glucosidase |
Ginkgolic Acid (C13:0) (6-Tridecylsalicylic acid): 0exhibits the highest α-glucosidase inhibitory activity. | |||
TN1705 | Glycyrrhisoflavone | MAO , Tyrosinase , NO Synthase , Immunology/Inflammation related | |
Glycyrrhisoflavone is a tyrosinase inhibitor with anti-inflammatory effects. Glycyrrhisoflavone inhibits α-glucosidase and monoamine oxidase. | |||
TN1928 | Methyl rosmarinate | MMP , Anti-infection , Tyrosinase | |
Methyl rosmarinate is a noncompetitive tyrosinase inhibitor which is isolated from Rabdosia serra, with an IC50 of 0.28 mM for mushroom tyrosinase.Methyl rosmarinate shows antioxidative, and antifungal activities. It has... | |||
T6S0535 | Pinoresinol diglucoside | Pinoresinol Diglucopyranoside | Glucosidase |
1. Pinoresinol diglucoside (Pinoresinol Diglucopyranoside) is a putative α-glucosidase inhibiting compound. 2. Pinoresinol diglucoside is a important antihypertensive compound. | |||
TN2277 | Torachrysone-8-O-b-D-glucoside | Torachrysone 8-O-glucoside | Antifection |
Torachrysone-8-O-b-D-glucoside shows alpha-glucosidase inhibitory activities, it may be used for the management of type 2 diabetes. | |||
TN2130 | Manghaslin | Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside | AChE , Glucosidase |
Manghaslin (Quercetin 3-O-rutinoside-(1->2)-O-rhamnoside) has considerable α-glucosidase inhibitory activity, illustrating the anti-diabetic potential of phenolic-rich litchi pulp extracts. Manghaslin also shows inhibito... | |||
T3796 | Betulinaldehyde | Betulinic aldehyde,Betulinal,Betunal | Apoptosis , Antibacterial |
Betulinaldehyde (Betunal) has the inhibition of Saccharomyces sp and alpha-glucosidase. Betulinaldehyde induces apoptosis in mouse B16 2F2 cells. Betulinaldehyde has anti-proliferative activity against mouse +SA mammary ... | |||
T6S1371 | Isovitexin | Homovitexin,Saponaretin,Apigenin-6-C-Glucoside | NF-κB , JNK , Glucosidase |
1. Isovitexin (Apigenin-6-C-Glucoside) exhibits a potential antioxidant activity. 2. Isovitexin shows a strong antihyperglycemic action, inhibits α-glucosidase in vivo. | |||
T5293 | Maltotriose | D-Maltotriose,Amylotriose | Others , Endogenous Metabolite |
Maltotriose (Amylotriose) is a common oligosaccharide metabolite found in human urine after maltose ingestion or infusion. Maltotriose is increased in Glycogen storage disease II due to a mutation of the enzyme alpha-1,4... | |||
T5690 | 7,4'-Di-O-methylapigenin | 4',7-DIMETHOXY-5-HYDROXYFLAVONE | Amylase |
7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) can inhibit α-glucosidase and α-amylase enzymes and enhance 2-NBDG uptake in L6 cells, it has hypolipidemic effect on mouse pre-adipocyte (3T3L1) cell lines. | |||
TN1956 | Mulberrofuran G | Phosphatase , HBV , Glucosidase | |
Mulberrofuran G, isolated from Morus alba L., has anti-hepatitis B virus activity and protects against ischemic injury-induced cell death. Mulberrofuran G is a dual inhibitor of PTP1B and alpha-glucosidase for use in the... | |||
TN4368 | Kaempferol-3,7-di-O-β-glucoside | Kaempferol 3,7-di-O-glucoside | Glucosidase , Amylase |
Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) is a flavonol from Morettia philaena, It can inhibit α-amylase, α-glucosidase and Acetylcholinesterase. Kaempferol-3, 7-di-o-β-Glucoside has neuroprotective ac... | |||
T5S1988 | Isorhamnetin-3-O-glucoside | Isorhamnetin-3-O-beta-D-Glucoside | Others |
Isorhamnetin-3-O-glucoside (Isorhamnetin-3-O-beta-D-Glucoside) inhibits the activity of alpha-glucosidase from rat intestine; it exhibits a potent rat lens aldose reductase (RLAR) inhibition in vitro, its IC(50) being 1.... | |||
T6S1369 | Vitexin | Apigenin-8-C-glucoside | Antioxidant |
1. Vitexin has antinociceptive and antispasmodic activities. 2. Vitexin exhibits a prominent first-pass effect. 3. Vitexin has antioxidant, antimyeloperoxidase, and α-glucosidase inhibitory activities. 4. Vitexin can eit... | |||
T2S0731 | Trilobatin | P-Phlorizin | Amylase |
Trilobatin (P-Phlorizin) has anti-oxidant effect, can increase superoxide dismutase (SOD) activity.Trilobatin has anti-inflammatory effect, it potentially inhibits the lipopolysaccharide (LPS)-induced inflammatory respon... | |||
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Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-05099 | GBA/glucocerebrosidase Protein, Human, Recombinant (His) | Human | HEK293 |
Mutations in the GBA gene, encoding the lysosomal hydrolase glucocerebrosidase (GCase), are the most common known genetic risk factor for Parkinson's disease (PD) and dementia with Lewy bodies (DLB). ASAH1 (acid ceramida... | |||
TMPY-01579 | GBA3 Protein, Human, Recombinant (His) | Human | Baculovirus-Insect Cells |
Cytosolic beta-glucosidase, also known as Cytosolic beta-glucosidase-like protein 1, GBA3, CBG and CBGL1 is a cytoplasm protein which belongs to theglycosyl hydrolase 1 family and Klotho subfamily. GBA3 / CBGL1 is a glyc... | |||
TMPH-03484 | Agn1 Protein, S. pombe, Recombinant (His & Myc) | Fission yeast | E. coli |
Has a role in cell separation where it is required for the degradation of the cell wall material surrounding the septum (the septum edging) which must be hydrolyzed before full separation of the daughter cells can occur.... |
Cat No. | Product Name | ||
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L7100 | Anti-Obesity Compound Library | 2286 compounds | |
A unique collection of 2286 anti-obesity compounds for high throughput and high content screening; |