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Search Result

Search Results for " glur "

Targets

iGluR GluR GluR

26

Compounds

2

Natural Products

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T9970 MGluR3 modulator-1 1-ethyl-3-(morpholin-4-yl)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile GluR
mGluR3 modulator-1 (1-ethyl-3-(morpholin-4-yl)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile) is a positive allosteric modulator of mGluR3 and can be used in studies about the treatment of Parkinson's disease.
T12717 Basimglurant CTEP Derivative,RG7090 GluR
Basimglurant (CTEP Derivative) is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd of 1.1 nM).
T35028 Valiglurax VU2957,VU 0652957,VU 2957,VU-0652957,VU0652957,VU-2957 GluR
Valiglurax (VU2957), also known as VU0652957 and VU2957, is a potent, selective, CNS penetrant, and orally bioavailable mGlu4 PAM. VU2957 possessed attractive in vitro and in vivo pharmacological and DMPK properties acro...
T15090 Decoglurant RO4995819 GluR
Decoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3 and it also is developed as an antidepressant.
T38612 Linaprazan glurate Others
Linaprazan glurate inhibits exogenously or endogenously stimulated gastric acid secretion. Linaprazan glurate can be used in studies about gastrointestinal inflammatory diseases and peptic ulcer diseases.
T9723 GluR6 antagonist-1 Src
GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.
T60882 MGluR2 modulator 2
mGluR2 modulator 2 (compound 2) can be used in antipsychotic research. mGluR2 modulator 2 is a potent, selective and orally bioavailable positive allosteric modulator of mGluR2 with an EC 50 value of 0.13 μM [1].
T15134 Dipraglurant ADX48621 Others
Dipraglurant is a negative allosteric regulator (NAM) of blood-brain barrier transmissible mGluR5 with effective, selective and oral activity, with an IC50 value of 21 nM. Dipraglurant can treat levodopa-induced dyskines...
T61277 MGluR2 modulator 4
mGluR2 modulator 4 (compound 47) is a highly potent positive allosteric modulator of mGluR2, exhibiting an EC 50 value of 0.8 μM. It holds the potential for investigating antipsychotic properties [1].
T34282 Remeglurant
Remeglurant is used as a selective antagonist of the mGlu5 receptor.
T11951 Mavoglurant racemate AFQ-056 racemate Others
Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.
T32080 Histidine oxoglurate Histidine alpha-ketoglutarate
Histidine oxoglurate is a bioactive chemical.
T82295 GluR23Y
GluR23Y, a biologically active peptide, was utilized in an ELISA-based cell-surface assay to assess insulin-stimulated endocytosis of native AMPA receptors in cultured hippocampal neurons. GluR23Y effectively inhibited t...
T80246 TAT-GluR23A Fusion Peptide
TAT-GluR23A Fusion Peptide is a bioactive peptide comprising the GluR23A sequence—residues 869 to 877 of GluR23Y with alanine replacing tyrosine—and an 11 amino acid cell-permeable HIV Trans-Activator of Transcription (T...
T38910 MGluR2 antagonist 1
mGluR2 antagonist 1 is a potent and selective class of negative allosteric modulator targeting the metabotropic glutamate receptor 2 (mGluR2) with high oral bioavailability. It displays a remarkable affinity for mGluR2, ...
T11311L Foliglurax PXT002331 GluR
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
T17241 Auglurant VU0424238 Others
Auglurant is a novel and selective mGlu5 antagonist (IC50: 11 nM (rat) and an IC50: 14 nM (human)). Auglurant has an acceptable CNS penetration.
T11311 Foliglurax monohydrochloride PXT002331 (monohydrochloride) Others
Foliglurax monohydrochloride Antiparkinsonian effect. is a highly selective and potent, brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) , with an EC50 of 79 nM.
T81801 MGluR5 antagonist-1
mGluR5 antagonist-1 (compound 10) is a potent mGluR5 inhibitor exhibiting an IC50 of 11.5 nM and demonstrates antidepressant effects [1].
T62202 MGluR2 modulator 1
mGluR2 modulator 1 (compound 95) is a potent, blood-brain-barrier permeable modulator of mGluR2 (metabotropic glutamate receptor-2) positive transmutation (EC50: 0.03 μM). mGluR2 modulator 1 can be used in the study of p...
T38659 MGluR5 modulator 1
mGluR5 modulator 1 is a compound that acts as a positive allosteric modulator of the metabotropic glutamate receptor subtype 5 (mGluR5). Its primary application lies in the field of schizophrenia and cognitive impairment...
T3486 3-MATIDA GluR , NMDAR
3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a). Displays ≥ 40-fold selectivity over other receptors: mGluR-5, mGluR-2, mGluR-4 (mGluR-4a) (IC50 > 300 μM), NMDA and GluR (AMPA) (IC50 = 250 μM). 3...
T6562 Latrepirdine dihydrochloride Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin Beta Amyloid , 5-HT Receptor , Adrenergic Receptor , GluR , Autophagy , Histamine Receptor
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug.
T14130 Adomeglivant LY2409021 Glucagon Receptor
Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
T81912 LSP-GR3 iGluR
LSP-GR3, a novel splice modulating oligomer (SMO) consisting of chemically-modified RNA oligonucleotides, potently and specifically directs the alternative splicing of GluR to promote GluR3-flip expression across the cen...
T76278 Efinopegdutide
Efinopegdutide (JNJ-64565111) is a potent dual agonist for the glucagon-like peptide-1 (GLP-1) and glucagon receptors (GluR), showing efficacy in activating both receptors. It has potential applications in the research o...

Compounds

mGluR3 modulator-1
T9970
Synonym: 1-ethyl-3-(morpholin-4-yl)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile
Target: GluR
Basimglurant
T12717
Synonym: CTEP Derivative,RG7090
Target: GluR
Valiglurax
T35028
Synonym: VU2957,VU 0652957,VU 2957,VU-0652957,VU0652957,VU-2957
Target: GluR
Decoglurant
T15090
Synonym: RO4995819
Target: GluR
Linaprazan glurate
T38612
Synonym:
Target: Others
GluR6 antagonist-1
T9723
Synonym:
Target: Src
mGluR2 modulator 2
T60882
Synonym:
Target:
Dipraglurant
T15134
Synonym: ADX48621
Target: Others
mGluR2 modulator 4
T61277
Synonym:
Target:
Remeglurant
T34282
Synonym:
Target:
Mavoglurant racemate
T11951
Synonym: AFQ-056 racemate
Target: Others
Histidine oxoglurate
T32080
Synonym: Histidine alpha-ketoglutarate
Target:
GluR23Y
T82295
Synonym:
Target:
TAT-GluR23A Fusion Peptide
T80246
Synonym:
Target:
mGluR2 antagonist 1
T38910
Synonym:
Target:
Foliglurax
T11311L
Synonym: PXT002331
Target: GluR
Auglurant
T17241
Synonym: VU0424238
Target: Others
Foliglurax monohydrochloride
T11311
Synonym: PXT002331 (monohydrochloride)
Target: Others
mGluR5 antagonist-1
T81801
Synonym:
Target:
mGluR2 modulator 1
T62202
Synonym:
Target:
mGluR5 modulator 1
T38659
Synonym:
Target:
3-MATIDA
T3486
Synonym:
Target: GluR, NMDAR
Latrepirdine dihydrochloride
T6562
Synonym: Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin
Target: Beta Amyloid, 5-HT Receptor, Adrenergic Receptor, GluR, Autophagy, Histamine Receptor
Adomeglivant
T14130
Synonym: LY2409021
Target: Glucagon Receptor
LSP-GR3
T81912
Synonym:
Target: iGluR
Efinopegdutide
T76278
Synonym:
Target:
Cat No. Product Name Synonyms Targets
T8626 Transtorine 1,4-DIHYDRO-4-OXOQUINOLINE-2-CARBOXYLIC ACID GluR , NMDAR
Transtorine (1,4-DIHYDRO-4-OXOQUINOLINE-2-CARBOXYLIC ACID) is a GluR and NMDA inhibitor.
T20191 (-)-Camphoric acid L-Camphoric acid,Camphoric acid, (-)- GluR
(-)-Camphoric acid (L-Camphoric acid) is a less active enantiomer of Camphoric acid which induces GluR expression.

Natural Products

Transtorine
T8626
Synonym: 1,4-DIHYDRO-4-OXOQUINOLINE-2-CARBOXYLIC ACID
Target: GluR, NMDAR
(-)-Camphoric acid
T20191
Synonym: L-Camphoric acid,Camphoric acid, (-)-
Target: GluR

Recombinant Proteins

Species：
Human (2)
Expression System：
E. coli (1)
HEK293 (1)
Tag：
His (1)
hFc (1)
Cat No. Product Name Species Expression System
TMPY-06701 GPX4 Protein, Human, Recombinant (His) Human E. coli
TMPY-04318 GRIK2 Protein, Human, Recombinant (hFc) Human HEK293
GRIK2 (Glutamate Ionotropic Receptor Kainate Type Subunit 2, also known as GluR6) is a Protein Coding gene. The GRIK2 (one of the kainate receptors) gene resides in a genetic linkage region (6q21) associated with bipolar...
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