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Mubritinib  
Catalog No. T6124    CAS 366017-09-6
Pack Size
Availability
Price/USD
Quantity
25mg
In stock
114.00
50mg
In stock
179.00
100mg
In stock
322.00
200mg
In stock
451.00
1 mL * 10 mM (in DMSO)
In stock
50.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.57% COA Datasheet HNMR HPLC
Biological Activity:

Product Description:

Mubritinib (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM.

Target:
PDGFR; JAK1; HER2/ErbB2; FGFR; EGFR;
Research Area:
Cancer
Chemical Information:
Molecular Weight 468.47
Formula C25H23F3N4O2
CAS Number 366017-09-6
Solubility DMSO:35.1 mg/mL (75 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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